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Design, Synthesis, and Biological Evaluation of Artemisinin-Indoloquinoline Hybrids as Potent Antiproliferative Agents

A series of artemisinin-indoloquinoline hybrids were designed and synthesized in an attempt to develop potent and selective anti-tumor agents. Compounds 7a–7f, 8 and 9 were prepared and characterized. Their antiproliferative activities against MV4-11, HCT-116, A549, and BALB/3T3 cell lines in vitro...

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Detalles Bibliográficos
Autores principales: Wang, Li, Świtalska, Marta, Wang, Ning, Du, Zhen-Jun, Fukumoto, Yuta, Diep, Nguyen Kim, Kiguchi, Ryo, Nokami, Junzo, Wietrzyk, Joanna, Inokuchi, Tsutomu
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2014
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6271626/
https://www.ncbi.nlm.nih.gov/pubmed/25412047
http://dx.doi.org/10.3390/molecules191119021