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Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action
Fungal pathogens continue to pose challenges to humans and plants despite efforts to control them. Two coumarins, robustic acid and thonningine-C isolated from Millettia thonningii, show promising activity against the fungus Candida albicans with minimum fungicidal concentration of 1.0 and 0.5 mg/mL...
Autores principales: | , , , , , , , , |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2016
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6274499/ https://www.ncbi.nlm.nih.gov/pubmed/27754464 http://dx.doi.org/10.3390/molecules21101369 |
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author | Ayine-Tora, Daniel M. Kingsford-Adaboh, Robert Asomaning, William A. Harrison, Jerry J.E.K. Mills-Robertson, Felix C. Bukari, Yahaya Sakyi, Patrick O. Kaminta, Sylvester Reynisson, Jóhannes |
author_facet | Ayine-Tora, Daniel M. Kingsford-Adaboh, Robert Asomaning, William A. Harrison, Jerry J.E.K. Mills-Robertson, Felix C. Bukari, Yahaya Sakyi, Patrick O. Kaminta, Sylvester Reynisson, Jóhannes |
author_sort | Ayine-Tora, Daniel M. |
collection | PubMed |
description | Fungal pathogens continue to pose challenges to humans and plants despite efforts to control them. Two coumarins, robustic acid and thonningine-C isolated from Millettia thonningii, show promising activity against the fungus Candida albicans with minimum fungicidal concentration of 1.0 and 0.5 mg/mL, respectively. Molecular modelling against the putative bio-molecular target, lanosterol 14α-demethylase (CYP51), revealed a plausible binding mode for the active compounds, in which the hydroxyl group binds with a methionine backbone carboxylic group blocking access to the iron catalytic site. This binding disrupts the synthesis of several important sterols for the survival of fungi. |
format | Online Article Text |
id | pubmed-6274499 |
institution | National Center for Biotechnology Information |
language | English |
publishDate | 2016 |
publisher | MDPI |
record_format | MEDLINE/PubMed |
spelling | pubmed-62744992018-12-28 Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action Ayine-Tora, Daniel M. Kingsford-Adaboh, Robert Asomaning, William A. Harrison, Jerry J.E.K. Mills-Robertson, Felix C. Bukari, Yahaya Sakyi, Patrick O. Kaminta, Sylvester Reynisson, Jóhannes Molecules Article Fungal pathogens continue to pose challenges to humans and plants despite efforts to control them. Two coumarins, robustic acid and thonningine-C isolated from Millettia thonningii, show promising activity against the fungus Candida albicans with minimum fungicidal concentration of 1.0 and 0.5 mg/mL, respectively. Molecular modelling against the putative bio-molecular target, lanosterol 14α-demethylase (CYP51), revealed a plausible binding mode for the active compounds, in which the hydroxyl group binds with a methionine backbone carboxylic group blocking access to the iron catalytic site. This binding disrupts the synthesis of several important sterols for the survival of fungi. MDPI 2016-10-15 /pmc/articles/PMC6274499/ /pubmed/27754464 http://dx.doi.org/10.3390/molecules21101369 Text en © 2016 by the authors. Licensee MDPI, Basel, Switzerland. This article is an open access article distributed under the terms and conditions of the Creative Commons Attribution (CC-BY) license (http://creativecommons.org/licenses/by/4.0/). |
spellingShingle | Article Ayine-Tora, Daniel M. Kingsford-Adaboh, Robert Asomaning, William A. Harrison, Jerry J.E.K. Mills-Robertson, Felix C. Bukari, Yahaya Sakyi, Patrick O. Kaminta, Sylvester Reynisson, Jóhannes Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action |
title | Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action |
title_full | Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action |
title_fullStr | Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action |
title_full_unstemmed | Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action |
title_short | Coumarin Antifungal Lead Compounds from Millettia thonningii and Their Predicted Mechanism of Action |
title_sort | coumarin antifungal lead compounds from millettia thonningii and their predicted mechanism of action |
topic | Article |
url | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6274499/ https://www.ncbi.nlm.nih.gov/pubmed/27754464 http://dx.doi.org/10.3390/molecules21101369 |
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