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Regioselective Synthesis of New 2,4-(Het)aryl-3H-pyrido[1′,2′:1,5]pyrazolo[4,3-d]pyrimidines Involving Palladium-Catalyzed Cross-Coupling Reactions

The design of some novel di-(het)arylated-3H-pyrido[1′,2′:1,5]pyrazolo[4,3-d]pyrimidine derivatives is reported. The series was developed from 1-aminopyridinium iodide, which afforded the key intermediate bearing two thiomethyl and amide functions, each of them useful for palladium catalyzed cross c...

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Detalles Bibliográficos
Autores principales:	Ejjoummany, Abdelaziz, Belaroussi, Rabia, El Hakmaoui, Ahmed, Akssira, Mohamed, Guillaumet, Gérald, Buron, Frédéric, Routier, Sylvain
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2018
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6278517/ https://www.ncbi.nlm.nih.gov/pubmed/30360579 http://dx.doi.org/10.3390/molecules23112740

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