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Synthesis of a benzoxazinthione derivative of tanaproget and pharmacological evaluation for PET imaging of PR expression

BACKGROUND: The histological evaluation of estrogen receptor (ER) and progesterone receptor (PR) expression in breast cancer lesions from biopsy tissue can stratify patients to receive endocrine therapy. Furthermore, PR expression can predict response to selective estrogen receptor modulators (SERMs...

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Detalles Bibliográficos
Autores principales:	Allott, Louis, Miranda, Cecilia, Hayes, Angela, Raynaud, Florence, Cawthorne, Christopher, Smith, Graham
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Springer International Publishing 2019
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6328429/ https://www.ncbi.nlm.nih.gov/pubmed/31659497 http://dx.doi.org/10.1186/s41181-018-0054-z

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