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Synthesis, Antibacterial and Antitubercular Activities of Some 5H-Thiazolo[3,2-a]pyrimidin-5-ones and Sulfonic Acid Derivatives

A series of 5H-thiazolo[3,2-a]pyrimidin-5-ones were synthesized by the cyclization reactions of S-alkylated derivatives in concentrated H(2)SO(4). Upon treatment of S-alkylated derivatives at different temperatures, intramolecular cyclization to 7-(substituted phenylamino)-5H-thiazolo[3,2-a]pyrimidi...

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Detalles Bibliográficos
Autores principales:	Cai, Dong, Zhang, Zhi-Hua, Chen, Yu, Yan, Xin-Jia, Zou, Liang-Jing, Wang, Ya-Xin, Liu, Xue-Qi
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2015
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6332143/ https://www.ncbi.nlm.nih.gov/pubmed/26378507 http://dx.doi.org/10.3390/molecules200916419

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