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Structure‐Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands(†)
New classes of alkylated hetarylpropylguanidines with different functionality and variation in spacer length were synthesized to determine their behavior at the four histamine receptor (H(1)R, H(2)R, H(3)R, H(4)R) subtypes. Alkylated guanidines with different terminal functional groups and varied ba...
Autores principales: | Pockes, Steffen, Wifling, David, Buschauer, Armin, Elz, Sigurd |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2019
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6401531/ https://www.ncbi.nlm.nih.gov/pubmed/30886786 http://dx.doi.org/10.1002/open.201900011 |
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