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Aromatic Bromination Abolishes the Psychomotor Features and Pro-social Responses of MDMA (“Ecstasy”) in Rats and Preserves Affinity for the Serotonin Transporter (SERT)

The entactogen MDMA (3,4-methylenedioxy-methamphetamine, “Ecstasy”) exerts its psychotropic effects acting primarily as a substrate of the serotonin transporter (SERT) to induce a non-exocytotic release of serotonin. Nevertheless, the roles of specific positions of the aromatic ring of MDMA associat...

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Detalles Bibliográficos
Autores principales:	Sáez-Briones, Patricio, Castro-Castillo, Vicente, Díaz-Véliz, Gabriela, Valladares, Luis, Barra, Rafael, Hernández, Alejandro, Cassels, Bruce K.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Frontiers Media S.A. 2019
Materias:	Pharmacology
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6403168/ https://www.ncbi.nlm.nih.gov/pubmed/30873030 http://dx.doi.org/10.3389/fphar.2019.00157

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