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Biased Signaling and Allosteric Modulation at the FSHR
Knowledge on G protein-coupled receptor (GPCRs) structure and mechanism of activation has profoundly evolved over the past years. The way drugs targeting this family of receptors are discovered and used has also changed. Ligands appear to bind a growing number of GPCRs in a competitive or allosteric...
Autores principales: | Landomiel, Flavie, De Pascali, Francesco, Raynaud, Pauline, Jean-Alphonse, Frédéric, Yvinec, Romain, Pellissier, Lucie P., Bozon, Véronique, Bruneau, Gilles, Crépieux, Pascale, Poupon, Anne, Reiter, Eric |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Frontiers Media S.A.
2019
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6425863/ https://www.ncbi.nlm.nih.gov/pubmed/30930853 http://dx.doi.org/10.3389/fendo.2019.00148 |
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