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Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
We designed and synthesised novel N-substituted 1,3-thiazolidin-4-one derivatives for the evaluation of their anti-Toxoplasma gondii efficacy. This scaffold was functionalised both at the N1-hydrazine portion with three structurally different moieties and at the lactam nitrogen with substituted benz...
Autores principales: | Carradori, Simone, Secci, Daniela, Bizzarri, Bruna, Chimenti, Paola, De Monte, Celeste, Guglielmi, Paolo, Campestre, Cristina, Rivanera, Daniela, Bordón, Claudia, Jones-Brando, Lorraine |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Taylor & Francis
2017
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6445228/ https://www.ncbi.nlm.nih.gov/pubmed/28537532 http://dx.doi.org/10.1080/14756366.2017.1316494 |
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