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Synthesis of New GABA(A) Receptor Modulator with Pyrazolo[1,5-a]quinazoline (PQ) Scaffold

We previously published a series of 8-methoxypirazolo[1,5-a]quinazolines (PQs) and their 4,5-dihydro derivatives (4,5(H)PQ) bearing the (hetero)arylalkylester group at position 3 as ligands at the γ-aminobutyric type A (GABA(A)) subtype receptor. Continuing the study in this field, we report here th...

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Detalles Bibliográficos
Autores principales:	Guerrini, Gabriella, Vergelli, Claudia, Cantini, Niccolò, Giovannoni, Maria Paola, Daniele, Simona, Mascia, Maria Paola, Martini, Claudia, Crocetti, Letizia
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2019
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6470557/ https://www.ncbi.nlm.nih.gov/pubmed/30901916 http://dx.doi.org/10.3390/ijms20061438

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