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Desulfonative photoredox alkylation of N-heteroaryl sulfones – an acid-free approach for substituted heteroarene synthesis
Minisci-type alkylation of electron-deficient heteroarenes has been a pivotal technique for medicinal chemists in the synthesis of drug-like molecules. However, such transformations usually require harsh conditions (e.g., strong acids, stoichiometric amount of oxidants, elevated temperatures, etc.)....
Autores principales: | Wang, Zheng-Jun, Zheng, Shuai, Matsui, Jennifer K., Lu, Zhipeng, Molander, Gary A. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Royal Society of Chemistry
2019
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6482881/ https://www.ncbi.nlm.nih.gov/pubmed/31057765 http://dx.doi.org/10.1039/c9sc00776h |
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