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Reactions of Piperazin-2-one, Morpholin-3-one, and Thiomorpholin-3-one with Triethyl Phosphite Prompted by Phosphoryl Chloride: Scope and Limitations
[Image: see text] The reaction of the title lactams with triethyl phosphite prompted by phosphoryl chloride provided six-membered ring heterocyclic phosphonates or bisphosphonates. These novel scaffolds might be of interest as building blocks in medicinal chemistry. The course of the reaction was de...
Autores principales: | Argüello-Velasco, Rubén Oswaldo, Dziuk, Błażej, Zarychta, Bartosz, Ordóñez, Mario, Kafarski, Paweł |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2019
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6648091/ https://www.ncbi.nlm.nih.gov/pubmed/31459993 http://dx.doi.org/10.1021/acsomega.9b01137 |
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