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Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamides as carbonic anhydrase isoforms I and II inhibitors

Carbonic anhydrases (CAs, EC 4.2.1.1) are crucial metalloenzymes that are involved in diverse bioprocesses. We report the synthesis and biological evaluation of novel series of benzenesulfonamides incorporating un/substituted ethyl quinoline-3-carboxylate moieties. The newly synthesised compounds we...

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Detalles Bibliográficos
Autores principales:	Al-Sanea, Mohammad M., Elkamhawy, Ahmed, Paik, Sora, Bua, Silvia, Ha Lee, So, Abdelgawad, Mohamed A., Roh, Eun Joo, Eldehna, Wagdy M., Supuran, Claudiu T.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2019
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6713088/ https://www.ncbi.nlm.nih.gov/pubmed/31411080 http://dx.doi.org/10.1080/14756366.2019.1652282

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