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Discovery of Novel Integrase Inhibitors Acting outside the Active Site Through High-Throughput Screening
Currently, an increasing number of drugs are becoming available to clinics for the treatment of HIV infection. Even if this targeted therapy is highly effective at suppressing viral replication, caregivers are facing growing therapeutic failures in patients, due to resistance with or without treatme...
Autores principales: | Aknin, Cindy, Smith, Elena A., Marchand, Christophe, Andreola, Marie-Line, Pommier, Yves, Metifiot, Mathieu |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2019
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6832134/ https://www.ncbi.nlm.nih.gov/pubmed/31614773 http://dx.doi.org/10.3390/molecules24203675 |
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