Cargando…

Phenylboronic Acids Probing Molecular Recognition against Class A and Class C β-lactamases

Worldwide dissemination of pathogens resistant to almost all available antibiotics represent a real problem preventing efficient treatment of infectious diseases. Among antimicrobial used in therapy, β-lactam antibiotics represent 40% thus playing a crucial role in the management of infections treat...

Descripción completa

Detalles Bibliográficos
Autores principales:	Linciano, Pasquale, Vicario, Mattia, Kekez, Ivana, Bellio, Pierangelo, Celenza, Giuseppe, Martín-Blecua, Isabel, Blázquez, Jesús, Cendron, Laura, Tondi, Donatella
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2019
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6963673/ https://www.ncbi.nlm.nih.gov/pubmed/31574990 http://dx.doi.org/10.3390/antibiotics8040171

Ejemplares similares

In silico identification and experimental validation of hits active against KPC-2 β-lactamase
por: Klein, Raphael, et al.
Publicado: (2018)

4-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases
por: Linciano, Pasquale, et al.
Publicado: (2020)

Targeting the Class A Carbapenemase GES-5 via Virtual Screening
por: Klein, Raphael, et al.
Publicado: (2020)

Targeting Class A and C Serine β-Lactamases with a Broad-Spectrum Boronic Acid Derivative
por: Tondi, Donatella, et al.
Publicado: (2014)

Protocetraric and Salazinic Acids as Potential Inhibitors of SARS-CoV-2 3CL Protease: Biochemical, Cytotoxic, and Computational Characterization of Depsidones as Slow-Binding Inactivators
por: Fagnani, Lorenza, et al.
Publicado: (2022)

New and simplified method for drug combination studies by checkerboard assay
por: Bellio, Pierangelo, et al.
Publicado: (2021)

Acquired Class D β-Lactamases
por: Antunes, Nuno T., et al.
Publicado: (2014)

Copper Binding and Oligomerization Studies of the Metal Resistance Determinant CrdA from Helicobacter pylori
por: Kekez, Ivana, et al.
Publicado: (2022)

Genomic analysis of bifunctional Class C-Class D β-lactamases in environmental bacteria
por: Silveira, Melise Chaves, et al.
Publicado: (2018)

Interaction of Avibactam with Class B Metallo-β-Lactamases
por: Abboud, Martine I., et al.
Publicado: (2016)

698. Nacubactam Inhibits Class A β-lactamases
por: Barnes, Melissa D, et al.
Publicado: (2018)

Intrinsic Class D β-Lactamases of Clostridium difficile
por: Toth, Marta, et al.
Publicado: (2018)

Cyclic Boronates Inhibit All Classes of β-Lactamases
por: Cahill, Samuel T., et al.
Publicado: (2017)

Salvianolic Acid B Strikes Back: New Evidence in the Modulation of Expression and Activity of Matrix Metalloproteinase 9 in MDA-MB-231 Human Breast Cancer Cells
por: Ianni, Andrea, et al.
Publicado: (2022)

Molecular Basis of Class A β-Lactamase Inhibition by Relebactam
por: Tooke, Catherine L., et al.
Publicado: (2019)

A Novel, Integron-Regulated, Class C β-Lactamase
por: Böhm, Maria-Elisabeth, et al.
Publicado: (2020)

The Role of Hydrophobic Nodes in the Dynamics of Class A β-Lactamases
por: Olehnovics, Edgar, et al.
Publicado: (2021)

Analysis of BlaEC family class C beta-lactamase
por: Schmidt, Jiri, et al.
Publicado: (2023)

Virtual screening identifies broad-spectrum β-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemases
por: Spyrakis, Francesca, et al.
Publicado: (2020)

Detection of Extended-Spectrum β-Lactamases (ESBLs) and AmpC in Class A and Class B Carbapenemase-Producing Enterobacterales
por: Imkamp, Frank, et al.
Publicado: (2022)

Computational and biological profile of boronic acids for the detection of bacterial serine- and metallo-β-lactamases
por: Santucci, Matteo, et al.
Publicado: (2017)

Class D β-lactamases do exist in Gram-positive bacteria
por: Toth, Marta, et al.
Publicado: (2015)

Interactions between Avibactam and Ceftazidime-Hydrolyzing Class D β-Lactamases
por: Frère, Jean-Marie, et al.
Publicado: (2020)

Structurally Related Liposomes Containing N-Oxide Surfactants: Physicochemical Properties and Evaluation of Antimicrobial Activity in Combination with Therapeutically Available Antibiotics
por: Battista, Sara, et al.
Publicado: (2022)

Lactobacillus sakei Pro-Bio65 Reduces TNF-α Expression and Upregulates GSH Content and Antioxidant Enzymatic Activities in Human Conjunctival Cells
por: Iorio, Roberto, et al.
Publicado: (2021)

Can We Exploit β-Lactamases Intrinsic Dynamics for Designing More Effective Inhibitors?
por: Gianquinto, Eleonora, et al.
Publicado: (2020)

A “turn-on” ESIPT fluorescence probe of 2-(aminocarbonyl)phenylboronic acid for the selective detection of Cu(ii)
por: Jiang, Dandan, et al.
Publicado: (2022)

Tackling the Antibiotic Resistance Caused by Class A β-Lactamases through the Use of β-Lactamase Inhibitory Protein
por: Eiamphungporn, Warawan, et al.
Publicado: (2018)

Transient disappearance of CD19(+)/CD5(+) B‐lymphocyte clone in peripheral blood in a patient with CLL during SARS‐CoV‐2‐related mild disease
por: Barnabei, Remo, et al.
Publicado: (2021)

An Extended Reservoir of Class-D Beta-Lactamases in Non-Clinical Bacterial Strains
por: Lupo, Valérian, et al.
Publicado: (2022)

The roles of highly conserved, non‐catalytic residues in class A β‐lactamases
por: Chikunova, Aleksandra, et al.
Publicado: (2022)

Antimycotic Activity of Ozonized Oil in Liposome Eye Drops against Candida spp.
por: Celenza, Giuseppe, et al.
Publicado: (2020)

Evaluation of the Analytical Performances of the Biolabo SOLEA 100 Optical Coagulometer and Comparison with the Stago STA-R MAX Analyser in the Determination of PT, APTT, and Fibrinogen
por: Bellio, Pierangelo, et al.
Publicado: (2022)

Recognition of AMP, ADP and ATP through Cooperative Binding by Cu(II) and Zn(II) Complexes Containing Urea and/or Phenylboronic Acid Moieties
por: Carreira-Barral, Israel, et al.
Publicado: (2018)

Interdomain flexibility and interfacial integrity of β-lactamase inhibitory protein (BLIP) modulate its binding to class A β-lactamases
por: Huang, Liwen, et al.
Publicado: (2021)

Phenylboronic acid derivative-modified (6,5) single-wall carbon nanotube probes for detecting glucose and hydrogen peroxide
por: Qiao, Yunfan, et al.
Publicado: (2019)

NMR Investigation of the Supramolecular Complex Formed by a Phenylboronic Acid-Ferrocene Electroactive Probe and Native or Derivatized β-Cyclodextrin
por: Cesari, Andrea, et al.
Publicado: (2022)

A selective hybrid fluorescent sensor for fructose detection based on a phenylboronic acid and BODIPY-based hydrophobicity probe
por: Kashiwazaki, Gengo, et al.
Publicado: (2022)

Non-catalytic-Region Mutations Conferring Transition of Class A β-Lactamases Into ESBLs
por: Cao, Thinh-Phat, et al.
Publicado: (2020)

Inhibition of Class A β-Lactamase (TEM-1) by Narrow Fractions of Humic Substances
por: Mikhnevich, Tatyana A., et al.
Publicado: (2021)

Cannot write session to /tmp/vufind_sessions/sess_s34aj4mkjpu5cgiik8nbrca7ve