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Synthesis and human carbonic anhydrase I, II, VA, and XII inhibition with novel amino acid–sulphonamide conjugates

A series of amino acid–sulphonamide conjugates was prepared through benzotriazole mediated coupling reactions and characterised by (1)H-NMR, (13)C-NMR, MS, and FTIR spectroscopic techniques as well as elemental analysis. The carbonic anhydrase (CA, EC 4.2.1.1) inhibitory activity of the new compound...

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Detalles Bibliográficos
Autores principales:	Küçükbay, Hasan, Buğday, Nesrin, Küçükbay, F. Zehra, Ageli, Andrea, Bartolucci, Gianluca, Supuran, Claudiu T.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2020
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6968503/ https://www.ncbi.nlm.nih.gov/pubmed/31914827 http://dx.doi.org/10.1080/14756366.2019.1710503

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