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Site‐Selective Late‐Stage Aromatic [(18)F]Fluorination via Aryl Sulfonium Salts
Site‐selective functionalization of C−H bonds in small complex molecules is a long‐standing challenge in organic chemistry. Herein, we report a broadly applicable and site‐selective aromatic C−H dibenzothiophenylation reaction. The conceptual advantage of this transformation is further demonstrated...
Autores principales: | Xu, Peng, Zhao, Da, Berger, Florian, Hamad, Aboubakr, Rickmeier, Jens, Petzold, Roland, Kondratiuk, Mykhailo, Bohdan, Kostiantyn, Ritter, Tobias |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2019
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7004179/ https://www.ncbi.nlm.nih.gov/pubmed/31697427 http://dx.doi.org/10.1002/anie.201912567 |
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