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Novel anti-inflammatory and analgesic agents: synthesis, molecular docking and in vivo studies
Twelve new derivatives of benzothiazole bearing benzenesulphonamide and carboxamide were synthesised and investigated for their in vivo anti-inflammatory, analgesic and ulcerogenic activities. Molecular docking showed an excellent binding interaction of the synthesised compounds with the receptors,...
Autores principales: | Ugwu, David Izuchukwu, Okoro, Uchechukwu Christopher, Ukoha, Pius Onyeoziri, Gupta, Astha, Okafor, Sunday N. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Taylor & Francis
2018
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7011796/ https://www.ncbi.nlm.nih.gov/pubmed/29372659 http://dx.doi.org/10.1080/14756366.2018.1426573 |
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