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Inhibition studies of Brucella suis β-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides

The two β-carbonic anhydrases (CAs, EC 4.2.1.1) from the pathogenic bacterium Brucella suis, BsuCA1 and BsuCA2, were investigated for their inhibition profile with a series of pyridine-3-sulphonamide derivatives incorporating 4-hetaryl moieties. BsuCA1 was effectively inhibited by these sulphonamide...

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Detalles Bibliográficos
Autores principales:	Monti, Simona Maria, Meccariello, Angela, Ceruso, Mariangela, Szafrański, Krzysztof, Sławiński, Jarosław, Supuran, Claudiu T.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2017
Materias:	Short Communication
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7011973/ https://www.ncbi.nlm.nih.gov/pubmed/29271264 http://dx.doi.org/10.1080/14756366.2017.1413097

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