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Benzimidazole derivatives endowed with potent antileishmanial activity
Two sets of benzimidazole derivatives were synthesised and tested in vitro for activity against promastigotes of Leishmania tropica and L. infantum. Most of the tested compounds resulted active against both Leishmania species, with IC(50) values in the low micromolar/sub-micromolar range. Among the...
Autores principales: | Tonelli, Michele, Gabriele, Elena, Piazza, Francesca, Basilico, Nicoletta, Parapini, Silvia, Tasso, Bruno, Loddo, Roberta, Sparatore, Fabio, Sparatore, Anna |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Taylor & Francis
2017
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7011974/ https://www.ncbi.nlm.nih.gov/pubmed/29233048 http://dx.doi.org/10.1080/14756366.2017.1410480 |
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