Cargando…

Design, Synthesis and Biological Evaluation of Benzo[D]Thiazole with Dimethylpyrazol Derivatives

A series of new benzothiazole derivatives containing dimethylpyrazole were synthesized and evaluated for their anticonvulsant activity, neurotoxicity and cytotoxicity by using the maximal electroshock (MES), rotarod neurotoxicity (TOX) and MTT colorimetric assay. Among the compounds studied, four co...

Descripción completa

Detalles Bibliográficos
Autores principales:	Liu, Dachuan, Cheng, Xiu, Wang, Ying
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	West Asia Organization for Cancer Prevention 2019
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7062998/ https://www.ncbi.nlm.nih.gov/pubmed/31759376 http://dx.doi.org/10.31557/APJCP.2019.20.11.3487

Ejemplares similares

Design, synthesis, and apoptosis-promoting effect evaluation of novel pyrazole with benzo[d]thiazole derivatives containing aminoguanidine units
por: Liu, Da Chuan, et al.
Publicado: (2019)

Design, synthesis and biological evaluation of benzo-[d]-imidazo-[2,1-b]-thiazole and imidazo-[2,1-b]-thiazole carboxamide triazole derivatives as antimycobacterial agents
por: Chitti, Surendar, et al.
Publicado: (2022)

2-[5-(Benzo[d]thiazol-2-yl)thiophen-2-yl]benzo[d]thiazole
por: Potgieter, Kim, et al.
Publicado: (2010)

Synthesis and biological evaluation of thiazole derivatives as LbSOD inhibitors
por: Brito, Camila C. Bitencourt, et al.
Publicado: (2018)

Synthesis and Ab Initio/DFT Studies on 2-(4-methoxyphenyl)benzo[d]thiazole
por: Arslan, Hakan, et al.
Publicado: (2007)

Design, synthesis, molecular docking studies and biological evaluation of thiazole carboxamide derivatives as COX inhibitors
por: Hawash, Mohammed, et al.
Publicado: (2023)

Synthesis and Biological Evaluation of Thiazole-Based Derivatives as Potential Acetylcholinesterase Inhibitors
por: Hemaida, Aya Y., et al.
Publicado: (2021)

Design, synthesis and biological evaluation of novel thiazole-naphthalene derivatives as potential anticancer agents and tubulin polymerisation inhibitors
por: Wang, Guangcheng, et al.
Publicado: (2021)

Syntheses of Benzo[d]Thiazol-2(3H)-One Derivatives and Their Antidepressant and Anticonvulsant Effects
por: Jin, Qinghao, et al.
Publicado: (2019)

DFT study on some polythiophenes containing benzo[d]thiazole and benzo[d]oxazole: structure and band gap
por: Vu Quoc, Trung, et al.
Publicado: (2021)

Design, synthesis and fungicidal activity of isothiazole–thiazole derivatives
por: Wu, Qi-Fan, et al.
Publicado: (2018)

Design, Synthesis and Biological Evaluation of New Imidazo[2,1-b]Thiazole Derivatives as Selective COX-2 Inhibitors
por: Shahrasbi, Mahsa, et al.
Publicado: (2018)

A Novel Class of Selective Acetylcholinesterase Inhibitors: Synthesis and Evaluation of (E)-2-(Benzo[d]thiazol-2-yl)-3-heteroarylacrylonitriles
por: de la Torre, Pedro, et al.
Publicado: (2012)

Synthesis and Biological Evaluation of Thiazole-Based Derivatives with Potential against Breast Cancer and Antimicrobial Agents
por: Pivovarova, Ekaterina, et al.
Publicado: (2022)

Synthesis, Biological Evaluation, and Molecular Docking Studies of Novel Isatin-Thiazole Derivatives as α-Glucosidase Inhibitors
por: Xie, Zhenzhen, et al.
Publicado: (2017)

Design, synthesis, and biological evaluation of thiazole/thiadiazole carboxamide scaffold-based derivatives as potential c-Met kinase inhibitors for cancer treatment
por: Nan, Xiang, et al.
Publicado: (2023)

Synthesis and Anticandidal Activity Evaluation of New Benzimidazole-Thiazole Derivatives
por: Kaplancıklı, Zafer Asım, et al.
Publicado: (2017)

Synthesis and biological evaluation of new derivatives of thieno-thiazole and dihydrothiazolo-thiazole scaffolds integrated with a pyrazoline nucleus as anticancer and multi-targeting kinase inhibitors
por: Othman, Ismail M. M., et al.
Publicado: (2021)

Synthesis and X-Ray Structure of [N,N-Bis(3,5-dimethylpyrazol-1-ylmethyl)-1-hydroxy-2-aminoethane](3,5-dimethylpyrazole) copper(II) dinitrate
por: Kodadi, Mohamed El, et al.
Publicado: (2003)

Synthesis, Characterization, and Biological Activity of a Novel Series of Benzo[4,5]imidazo[2,1-b]thiazole Derivatives as Potential Epidermal Growth Factor Receptor Inhibitors
por: Deng, Xinshan, et al.
Publicado: (2019)

Synthesis, Structural Characterization, and Cytotoxic Activity of New Benzo[d]imidazo[2,1-b]thiazole Derivatives Against MCF-7 Breast Cancer Cells
por: Ahmadi, Nahid, et al.
Publicado: (2022)

3-(Benzo[d]thiazol-2-yl)-2H-chromen-2-one
por: Abdallah, Amira E. M., et al.
Publicado: (2022)

Design, Synthesis, and Biological Evaluation of Novel 6H-Benzo[c]chromen-6-one Derivatives as Potential Phosphodiesterase II Inhibitors
por: Tang, Long, et al.
Publicado: (2021)

Synthesis of N-(6-Arylbenzo[d]thiazole-2-acetamide Derivatives and Their Biological Activities: An Experimental and Computational Approach
por: Gull, Yasmeen, et al.
Publicado: (2016)

Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides
por: Abdoli, Morteza, et al.
Publicado: (2017)

(3,5-Dimethylpyrazol-1-yl)[5-(3,5-dimethylpyrazol-1-ylcarbonyl)-2-thienyl]methanone
por: Guzei, Ilia A., et al.
Publicado: (2009)

Synthesis and Anti-TMV Activity of Dialkyl/dibenzyl 2-((6-Substituted-benzo[d]thiazol-2-ylamino)(benzofuran-2-yl)methyl) Malonates
por: Xiao, Han, et al.
Publicado: (2013)

Synthesis, in silico studies and biological screening of (E)-2-(3-(substitutedstyryl)-5-(substitutedphenyl)-4,5-dihydropyrazol-1-yl)benzo[d]thiazole derivatives as an anti-oxidant, anti-inflammatory and antimicrobial agents
por: Kumar, Manoj, et al.
Publicado: (2022)

Synthesis, DFT Studies, Molecular Docking and Biological Activity Evaluation of Thiazole-Sulfonamide Derivatives as Potent Alzheimer’s Inhibitors
por: Khan, Shoaib, et al.
Publicado: (2023)

Synthesis, Structure and Molecular Docking of New 4,5-Dihydrothiazole Derivatives Based on 3,5-Dimethylpyrazole and Cytisine and Salsoline Alkaloids
por: Ibrayev, Marat K., et al.
Publicado: (2022)

Tackling Microbial Resistance with Isatin-Decorated Thiazole Derivatives: Design, Synthesis, and in vitro Evaluation of Antimicrobial and Antibiofilm Activity
por: Kassab, Refaie M, et al.
Publicado: (2022)

Synthesis and Anticancer Evaluation of New Thiazole and Thiadiazole Derivatives Bearing Acetanilide Moiety
por: El-Rayyes, Ali, et al.
Publicado: (2022)

One-Pot Chemoenzymatic Multicomponent Synthesis of Thiazole Derivatives
por: Zheng, Hui, et al.
Publicado: (2013)

Stereoselective synthesis, X-ray analysis, computational studies and biological evaluation of new thiazole derivatives as potential anticancer agents
por: Mabkhot, Yahia N., et al.
Publicado: (2018)

Butyl 3-oxo-2,3-dihydrobenzo[d][1,2]thiazole-2-carboxylate
por: Yang, Jian-Xin, et al.
Publicado: (2011)

Synthesis, Structure and Antifungal Activity of New 3-[(5-Aryl-1,3,4-oxadiazol-2-yl)methyl]benzo[d]thiazol-2(3H)-ones
por: Weng, Jian-Quan, et al.
Publicado: (2012)

2-(Benzo[d]thiazol-2-ylsulfonyl)-1-(4-bromophenyl)ethanone
por: Loghmani-Khouzani, Hossein, et al.
Publicado: (2009)

Crystal structure of 2-(2,5-dimethoxyphenyl)benzo[d]thiazole
por: Metwally, Nadia H., et al.
Publicado: (2022)

2-((1H-Benzo[d]imidazol-2-yl)amino)benzo[d]thiazole-6-sulphonamides: a class of carbonic anhydrase II and VII-selective inhibitors
por: Abdoli, Morteza, et al.
Publicado: (2023)

N-[(3,5-Dimethylpyrazol-1-yl)methyl]phthalimide
por: Wang, Su-Qing, et al.
Publicado: (2008)

Cannot write session to /tmp/vufind_sessions/sess_cs05cdc7h9at73c1flogdpccvm