Cargando…

The influence of ABCG2 polymorphism on erlotinib efflux in the K562 cell line

Single nucleotide polymorphisms (SNPs) in the gene for multidrug resistance protein ABCG2, an erlotinib transporter, is a possible contributor to the interindividual variation observed in erlotinib pharmacokinetics and toxicity. Therefore, the aim was to study erlotinib efflux by ABCG2 wild‐type (wt...

Descripción completa

Detalles Bibliográficos
Autores principales:	Svedberg, Anna, Jacobs, Lianne, Vikingsson, Svante, Gréen, Henrik
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2020
Materias:	Original Articles
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7138917/ https://www.ncbi.nlm.nih.gov/pubmed/32266784 http://dx.doi.org/10.1002/prp2.581

Ejemplares similares

Effect of ABCG2/BCRP Expression on Efflux and Uptake of Gefitinib in NSCLC Cell Lines
por: Galetti, Maricla, et al.
Publicado: (2015)

Celecoxib Up Regulates the Expression of Drug Efflux Transporter ABCG2 in Breast Cancer Cell Lines
por: Kalalinia, Fatemeh, et al.
Publicado: (2014)

Circumstances, Postmortem Findings, Blood Concentrations and Metabolism in a Series of Methoxyacetylfentanyl-Related Deaths
por: Kronstrand, Robert, et al.
Publicado: (2021)

AhR-activating pesticides increase the bovine ABCG2 efflux activity in MDCKII-bABCG2 cells
por: Kuhnert, Lydia, et al.
Publicado: (2020)

Molecular basis of cholesterol efflux via ABCG subfamily transporters
por: Sun, Yingyuan, et al.
Publicado: (2021)

Bioluminescent imaging of ABCG2 efflux activity at the blood-placenta barrier
por: Kumar, Jeyan S., et al.
Publicado: (2016)

Correlations between metabolism and structural elements of the alicyclic fentanyl analogs cyclopropyl fentanyl, cyclobutyl fentanyl, cyclopentyl fentanyl, cyclohexyl fentanyl and 2,2,3,3-tetramethylcyclopropyl fentanyl studied by human hepatocytes and LC-QTOF-MS
por: Åstrand, Anna, et al.
Publicado: (2018)

Characterization of an Etoposide‐resistant Human K562 Cell Line, K/eto
por: Sugawara, Isamu, et al.
Publicado: (1991)

Activation of the μ‐opioid receptor by alicyclic fentanyls: Changes from high potency full agonists to low potency partial agonists with increasing alicyclic substructure
por: Åstrand, Anna, et al.
Publicado: (2020)

RAGE Suppresses ABCG1-Mediated Macrophage Cholesterol Efflux in Diabetes
por: Daffu, Gurdip, et al.
Publicado: (2015)

Potential role of the ABCG2-Q141K polymorphism in type 2 diabetes
por: Szabó, Edit, et al.
Publicado: (2021)

Vorinostat enhances chemosensitivity to arsenic trioxide in K562 cell line
por: Li, Nainong, et al.
Publicado: (2015)

Simple and cost-effective liquid chromatography-mass spectrometry method to measure dabrafenib quantitatively and six metabolites semi-quantitatively in human plasma
por: Vikingsson, Svante, et al.
Publicado: (2017)

ABCG5 and ABCG8 Are Involved in Vitamin K Transport
por: Matsuo, Michinori, et al.
Publicado: (2023)

Structural basis for abscisic acid efflux mediated by ABCG25 in Arabidopsis thaliana
por: Ying, Wei, et al.
Publicado: (2023)

SR-BI associates with ABCG1 and inhibits ABCG1-mediated cholesterol efflux from cells to high-density lipoprotein 3
por: Song, Guohua, et al.
Publicado: (2012)

Metabolite Profiling of Ortho-, Meta- and Para-Fluorofentanyl by Hepatocytes and High-Resolution Mass Spectrometry
por: Gundersen, Per Ole M, et al.
Publicado: (2019)

Different toxic effects of YTX in tumor K-562 and lymphoblastoid cell lines
por: Fernández-Araujo, Andrea, et al.
Publicado: (2015)

Genomic amplification of chromosome 7 in the Doxorubicin resistant K562 cell line
por: Ibrahim, Sara.M, et al.
Publicado: (2018)

Mesalazine induces apoptosis via mitochondrial pathway in K562 cell line
por: Forsati, Parisa, et al.
Publicado: (2022)

Poziotinib Inhibits the Efflux Activity of the ABCB1 and ABCG2 Transporters and the Expression of the ABCG2 Transporter Protein in Multidrug Resistant Colon Cancer Cells
por: Zhang, Yongchao, et al.
Publicado: (2020)

ABCB1 1199G>A Genetic Polymorphism (Rs2229109) Influences the Intracellular Accumulation of Tacrolimus in HEK293 and K562 Recombinant Cell Lines
por: Dessilly, Géraldine, et al.
Publicado: (2014)

In Vitro Antileukemia Activity of ZSTK474 on K562 and Multidrug Resistant K562/A02 Cells
por: Zhou, Qianxiang, et al.
Publicado: (2016)

Extra-Renal Elimination of Uric Acid via Intestinal Efflux Transporter BCRP/ABCG2
por: Hosomi, Atsushi, et al.
Publicado: (2012)

ABCG2 is not able to catalyze glutathione efflux and does not contribute to GSH-dependent collateral sensitivity
por: Gauthier, Charlotte, et al.
Publicado: (2013)

Estrogen induces cell proliferation by promoting ABCG2-mediated efflux in endometrial cancer cells
por: Yaguchi, Takahiro, et al.
Publicado: (2018)

CM082 Enhances the Efficacy of Chemotherapeutic Drugs by Inhibiting the Drug Efflux Function of ABCG2
por: Xu, Lejia, et al.
Publicado: (2019)

CM082 Enhances the Efficacy of Chemotherapeutic Drugs by Inhibiting the Drug Efflux Function of ABCG2
por: Xu, Lejia, et al.
Publicado: (2023)

Effects of acceptor composition and mechanism of ABCG1-mediated cellular free cholesterol efflux
por: Sankaranarayanan, Sandhya, et al.
Publicado: (2009)

Correction: ABCB1 1199G>A Genetic Polymorphism (Rs2229109) Influences the Intracellular Accumulation of Tacrolimus in HEK293 and K562 Recombinant Cell Lines
Publicado: (2014)

Dexrazoxane significantly impairs the induction of doxorubicin resistance in the human leukaemia line, K562
por: Sargent, J M, et al.
Publicado: (2001)

Impairment of Methotrexate (MTX)‐Polyglutamate Formation of MTX‐resistant K562 Cell Lines
por: Koizumi, Shoichi
Publicado: (1988)

Effect of Chicken Bone Extracts on Metabolic and Mitochondrial Functions of K562 Cell Line
por: Pacelli, Consiglia, et al.
Publicado: (2020)

Proteomic Analysis of Quercetin-Treated K562 Cells
por: Brisdelli, Fabrizia, et al.
Publicado: (2019)

Rheumatoid Arthritis Disease Activity Is Determinant for ABCB1 and ABCG2 Drug-Efflux Transporters Function
por: Atisha-Fregoso, Yemil, et al.
Publicado: (2016)

Impact of cellular folate status and epidermal growth factor receptor expression on BCRP/ABCG2-mediated resistance to gefitinib and erlotinib
por: Lemos, C, et al.
Publicado: (2009)

Enhanced anti-proliferative action of busulphan by quercetin on the human leukaemia cell line K562.
por: Hoffman, R., et al.
Publicado: (1989)

Differential Gene Expression Analysis in K562 Human Leukemia Cell Line Treated with Benzene
por: Choi, Sulji, et al.
Publicado: (2011)

Kinetics of Internalization and Cytotoxicity of Transferrin‐Neocarzinostatin Conjugate in Human Leukemia Cell Line, K562
por: Kohgo, Yutaka, et al.
Publicado: (1990)

Comprehensive, integrated, and phased whole-genome analysis of the primary ENCODE cell line K562
por: Zhou, Bo, et al.
Publicado: (2019)

Cannot write session to /tmp/vufind_sessions/sess_5hn7vl3s11hfsch4gg1sn1aqco