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Development of Novel (111)-In-Labelled DOTA Urotensin II Analogues for Targeting the UT Receptor Overexpressed in Solid Tumours
Overexpression of G protein-coupled receptors (GPCRs) in tumours is widely used to develop GPCR-targeting radioligands for solid tumour imaging in the context of diagnosis and even treatment. The human vasoactive neuropeptide urotensin II (hUII), which shares structural analogies with somatostatin,...
Autores principales: | Poret, Benjamin, Desrues, Laurence, Bonin, Marc-André, Pedard, Martin, Dubois, Martine, Leduc, Richard, Modzelewski, Romain, Decazes, Pierre, Morin, Fabrice, Vera, Pierre, Castel, Hélène, Bohn, Pierre, Gandolfo, Pierrick |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7175314/ https://www.ncbi.nlm.nih.gov/pubmed/32204509 http://dx.doi.org/10.3390/biom10030471 |
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