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Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety
New dipeptide–dihydroquinolinone derivatives were successfully synthesised by benzotriazole mediated nucleophilic acyl substitution reaction and their structures were elucidated by spectroscopic and analytic techniques. The carbonic anhydrase (CA, EC 4.2.1.1) inhibitory activity of the new compounds...
Autores principales: | Küçükbay, Hasan, Gönül, Zeynep, Küçükbay, F. Zehra, Angeli, Andrea, Bartolucci, Gianluca, Supuran, Claudiu T. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Taylor & Francis
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7178833/ https://www.ncbi.nlm.nih.gov/pubmed/32297533 http://dx.doi.org/10.1080/14756366.2020.1751620 |
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