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Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling

1-[tert-Butyl(diphenyl)silyl]pyrrol-3-ylboronic acid was obtained from pyrrole in three steps. Its Suzuki–Miyaura cross-coupling with functionalized pyridinyl and pyrimidinyl bromides afforded new promising 3-hetaryl-1H-pyrroles.

Detalles Bibliográficos
Autores principales: Matyugina, Elena S., Khandazhinskaya, Anastasia L., Kochetkov, Sergey N., Seley-Radtke, Katherine L.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: 2020
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7241993/
http://dx.doi.org/10.1016/j.mencom.2020.03.034
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author Matyugina, Elena S.
Khandazhinskaya, Anastasia L.
Kochetkov, Sergey N.
Seley-Radtke, Katherine L.
author_facet Matyugina, Elena S.
Khandazhinskaya, Anastasia L.
Kochetkov, Sergey N.
Seley-Radtke, Katherine L.
author_sort Matyugina, Elena S.
collection PubMed
description 1-[tert-Butyl(diphenyl)silyl]pyrrol-3-ylboronic acid was obtained from pyrrole in three steps. Its Suzuki–Miyaura cross-coupling with functionalized pyridinyl and pyrimidinyl bromides afforded new promising 3-hetaryl-1H-pyrroles.
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spelling pubmed-72419932020-05-22 Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling Matyugina, Elena S. Khandazhinskaya, Anastasia L. Kochetkov, Sergey N. Seley-Radtke, Katherine L. Mendeleev Communications Article 1-[tert-Butyl(diphenyl)silyl]pyrrol-3-ylboronic acid was obtained from pyrrole in three steps. Its Suzuki–Miyaura cross-coupling with functionalized pyridinyl and pyrimidinyl bromides afforded new promising 3-hetaryl-1H-pyrroles. 2020 2020-05-21 /pmc/articles/PMC7241993/ http://dx.doi.org/10.1016/j.mencom.2020.03.034 Text en . Since January 2020 Elsevier has created a COVID-19 resource centre with free information in English and Mandarin on the novel coronavirus COVID-19. The COVID-19 resource centre is hosted on Elsevier Connect, the company's public news and information website. Elsevier hereby grants permission to make all its COVID-19-related research that is available on the COVID-19 resource centre - including this research content - immediately available in PubMed Central and other publicly funded repositories, such as the WHO COVID database with rights for unrestricted research re-use and analyses in any form or by any means with acknowledgement of the original source. These permissions are granted for free by Elsevier for as long as the COVID-19 resource centre remains active.
spellingShingle Article
Matyugina, Elena S.
Khandazhinskaya, Anastasia L.
Kochetkov, Sergey N.
Seley-Radtke, Katherine L.
Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling
title Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling
title_full Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling
title_fullStr Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling
title_full_unstemmed Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling
title_short Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling
title_sort synthesis of 3-hetarylpyrroles by suzuki–miyaura cross-coupling
topic Article
url https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7241993/
http://dx.doi.org/10.1016/j.mencom.2020.03.034
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