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Cell-Based Radiotracer Binding and Uptake Inhibition Assays: A Comparison of In Vitro Methods to Assess the Potency of Drugs That Target Monoamine Transporters
High-affinity monoamine transporters are targets for prescribed medications and stimulant drugs of abuse. Therefore, assessing monoamine transporter activity for candidate medications and newly-emerging drugs of abuse provides essential information for industry, academia, and public health. Radiotra...
Autores principales: | Ilic, Marija, Maier, Julian, Holy, Marion, Jaentsch, Kathrin, Liechti, Matthias E., Lubec, Gert, Baumann, Michael H., Sitte, Harald H., Luethi, Dino |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Frontiers Media S.A.
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7248194/ https://www.ncbi.nlm.nih.gov/pubmed/32508638 http://dx.doi.org/10.3389/fphar.2020.00673 |
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