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Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase
The ongoing Corona Virus Disease 2019 (COVID-19) pandemic, caused by severe acute respiratory syndrome coronavirus-2 (SARS-CoV-2), has emphasized the urgent need for antiviral therapeutics. The viral RNA-dependent-RNA-polymerase (RdRp) is a promising target with polymerase inhibitors successfully us...
Autores principales: | , , , , , , , , , , , , |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Cold Spring Harbor Laboratory
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7263509/ https://www.ncbi.nlm.nih.gov/pubmed/32511380 http://dx.doi.org/10.1101/2020.05.15.098731 |
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author | Shannon, A. Selisko, B. Le, NTT Huchting, J. Touret, F. Piorkowski, G. Fattorini, V. Ferron, F. Decroly, E. Meier, C Coutard, B. Peersen, O. Canard, B. |
author_facet | Shannon, A. Selisko, B. Le, NTT Huchting, J. Touret, F. Piorkowski, G. Fattorini, V. Ferron, F. Decroly, E. Meier, C Coutard, B. Peersen, O. Canard, B. |
author_sort | Shannon, A. |
collection | PubMed |
description | The ongoing Corona Virus Disease 2019 (COVID-19) pandemic, caused by severe acute respiratory syndrome coronavirus-2 (SARS-CoV-2), has emphasized the urgent need for antiviral therapeutics. The viral RNA-dependent-RNA-polymerase (RdRp) is a promising target with polymerase inhibitors successfully used for the treatment of several viral diseases. Here we show that Favipiravir exerts an antiviral effect as a nucleotide analogue through a combination of chain termination, slowed RNA synthesis and lethal mutagenesis. The SARS-CoV RdRp complex is at least 10-fold more active than any other viral RdRp known. It possesses both unusually high nucleotide incorporation rates and high-error rates allowing facile insertion of Favipiravir into viral RNA, provoking C-to-U and G-to-A transitions in the already low cytosine content SARS-CoV-2 genome. The coronavirus RdRp complex represents an Achilles heel for SARS-CoV, supporting nucleoside analogues as promising candidates for the treatment of COVID-19. |
format | Online Article Text |
id | pubmed-7263509 |
institution | National Center for Biotechnology Information |
language | English |
publishDate | 2020 |
publisher | Cold Spring Harbor Laboratory |
record_format | MEDLINE/PubMed |
spelling | pubmed-72635092020-06-07 Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase Shannon, A. Selisko, B. Le, NTT Huchting, J. Touret, F. Piorkowski, G. Fattorini, V. Ferron, F. Decroly, E. Meier, C Coutard, B. Peersen, O. Canard, B. bioRxiv Article The ongoing Corona Virus Disease 2019 (COVID-19) pandemic, caused by severe acute respiratory syndrome coronavirus-2 (SARS-CoV-2), has emphasized the urgent need for antiviral therapeutics. The viral RNA-dependent-RNA-polymerase (RdRp) is a promising target with polymerase inhibitors successfully used for the treatment of several viral diseases. Here we show that Favipiravir exerts an antiviral effect as a nucleotide analogue through a combination of chain termination, slowed RNA synthesis and lethal mutagenesis. The SARS-CoV RdRp complex is at least 10-fold more active than any other viral RdRp known. It possesses both unusually high nucleotide incorporation rates and high-error rates allowing facile insertion of Favipiravir into viral RNA, provoking C-to-U and G-to-A transitions in the already low cytosine content SARS-CoV-2 genome. The coronavirus RdRp complex represents an Achilles heel for SARS-CoV, supporting nucleoside analogues as promising candidates for the treatment of COVID-19. Cold Spring Harbor Laboratory 2020-05-15 /pmc/articles/PMC7263509/ /pubmed/32511380 http://dx.doi.org/10.1101/2020.05.15.098731 Text en http://creativecommons.org/licenses/by-nd/4.0/It is made available under a CC-BY-ND 4.0 International license (http://creativecommons.org/licenses/by-nd/4.0/) . |
spellingShingle | Article Shannon, A. Selisko, B. Le, NTT Huchting, J. Touret, F. Piorkowski, G. Fattorini, V. Ferron, F. Decroly, E. Meier, C Coutard, B. Peersen, O. Canard, B. Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase |
title | Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase |
title_full | Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase |
title_fullStr | Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase |
title_full_unstemmed | Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase |
title_short | Favipiravir strikes the SARS-CoV-2 at its Achilles heel, the RNA polymerase |
title_sort | favipiravir strikes the sars-cov-2 at its achilles heel, the rna polymerase |
topic | Article |
url | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7263509/ https://www.ncbi.nlm.nih.gov/pubmed/32511380 http://dx.doi.org/10.1101/2020.05.15.098731 |
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