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Isonitrile-Based Multicomponent Synthesis of β-Amino Boronic Acids as β-Lactamase Inhibitors

The application of various isonitrile-based multicomponent reactions to protected (2-oxoethyl)boronic acid (as the carbonyl component) is described. The Ugi reaction, both in the four components and in the four centers–three components versions, and the van Leusen reaction, proved effective at provi...

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Detalles Bibliográficos
Autores principales:	Bassini, Emanuele, Gazzotti, Stefano, Sannio, Filomena, Lo Presti, Leonardo, Sgrignani, Jacopo, Docquier, Jean-Denis, Grazioso, Giovanni, Silvani, Alessandra
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2020
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7277116/ https://www.ncbi.nlm.nih.gov/pubmed/32408714 http://dx.doi.org/10.3390/antibiotics9050249

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