B(C(6)F(5))(3)-Catalyzed Direct C3 Alkylation of Indoles and Oxindoles

[Image: see text] The direct C3 alkylation of indoles and oxindoles is a challenging transformation, and only a few direct methods exist. Utilizing the underexplored ability of triaryl boranes to mediate the heterolytic cleavage of α-nitrogen C–H bonds in amines, we have developed a catalytic approa...

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Detalles Bibliográficos
Autores principales: Basak, Shyam, Alvarez-Montoya, Ana, Winfrey, Laura, Melen, Rebecca L., Morrill, Louis C., Pulis, Alexander P.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2020
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7311048/
https://www.ncbi.nlm.nih.gov/pubmed/32596025
http://dx.doi.org/10.1021/acscatal.0c01141

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7311048/
https://www.ncbi.nlm.nih.gov/pubmed/32596025
http://dx.doi.org/10.1021/acscatal.0c01141

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