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Functional characterization of the antiepileptic drug candidate, padsevonil, on GABA(A) receptors

OBJECTIVE: The antiepileptic drug candidate, padsevonil, is the first in a novel class of drugs designed to interact with both presynaptic and postsynaptic therapeutic targets: synaptic vesicle 2 proteins and γ‐aminobutyric acid type A receptors (GABA(A)Rs), respectively. Functional aspects of padse...

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Detalles Bibliográficos
Autores principales:	Niespodziany, Isabelle, Ghisdal, Philippe, Mullier, Brice, Wood, Martyn, Provins, Laurent, Kaminski, Rafal M., Wolff, Christian
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2020
Materias:	Full‐length Original Research
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7383892/ https://www.ncbi.nlm.nih.gov/pubmed/32297665 http://dx.doi.org/10.1111/epi.16497

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