Cargando…

Physical stability and release properties of lumefantrine amorphous solid dispersion granules prepared by a simple solvent evaporation approach

Amorphous solid dispersions (ASDs) of lumefantrine, which has low aqueous solubility, have been shown to improve bioavailability relative to crystalline formulations. Herein, the crystallization tendency and release properties of a variety of lumefantrine ASD granules, formed on a blend of microcrys...

Descripción completa

Detalles Bibliográficos
Autores principales:	Trasi, Niraj S., Bhujbal, Sonal V., Zemlyanov, Dmitry Y., Zhou, Qi (Tony), Taylor, Lynne S.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Elsevier 2020
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7390794/ https://www.ncbi.nlm.nih.gov/pubmed/32760909 http://dx.doi.org/10.1016/j.ijpx.2020.100052

Ejemplares similares

Amorphous solid dispersion formation via solvent granulation – A case study with ritonavir and lopinavir
por: Trasi, Niraj S., et al.
Publicado: (2019)

Physical Stability and Dissolution of Lumefantrine Amorphous Solid Dispersions Produced by Spray Anti-Solvent Precipitation
por: Bhujbal, Sonal V., et al.
Publicado: (2021)

Effect of Storage Humidity on Physical Stability of Spray-Dried Naproxen Amorphous Solid Dispersions with Polyvinylpyrrolidone: Two Fluid Nozzle vs. Three Fluid Nozzle
por: Bhujbal, Sonal V., et al.
Publicado: (2021)

Pharmaceutical amorphous solid dispersion: A review of manufacturing strategies
por: Bhujbal, Sonal V., et al.
Publicado: (2021)

Water-Induced Phase Separation of Spray-Dried Amorphous Solid Dispersions
por: Li, Na, et al.
Publicado: (2020)

Molecular Disorder of Bicalutamide—Amorphous Solid Dispersions Obtained by Solvent Methods
por: Szafraniec, Joanna, et al.
Publicado: (2018)

Development, characterization and solubility study of solid dispersions of Cefuroxime Axetil by the solvent evaporation method
por: Arora, S. C., et al.
Publicado: (2010)

DEVELOPMENT, CHARACTERIZATION AND SOLUBILITY STUDY OF SOLID DISPERSIONS OF AZITHROMYCIN DIHYDRATE BY SOLVENT EVAPORATION METHOD
por: Arora, S.C., et al.
Publicado: (2010)

Solubility Improvement of Progesterone from Solid Dispersions Prepared by Solvent Evaporation and Co-milling
por: Chen, Xing, et al.
Publicado: (2020)

Solid-state characterization of lacidipine/PVP K(29/32) solid dispersion primed by solvent co-evaporation
por: Mukharya, Amit, et al.
Publicado: (2012)

Dissolution enhancement of glibenclamide by solid dispersion: solvent evaporation versus a supercritical fluid-based solvent -antisolvent technique
por: Tabbakhian, M., et al.
Publicado: (2014)

Improved dissolution of Kaempferia parviflora extract for oral administration by preparing solid dispersion via solvent evaporation
por: Weerapol, Yotsanan, et al.
Publicado: (2017)

Thermal Stability of Amorphous Solid Dispersions
por: Jelić, Dijana
Publicado: (2021)

Explaining the Release Mechanism of Ritonavir/PVPVA Amorphous Solid Dispersions
por: Krummnow, Adrian, et al.
Publicado: (2022)

Characterization of Amorphous Solid Dispersion of Pharmaceutical Compound with pH-Dependent Solubility Prepared by Continuous-Spray Granulator
por: Tanaka, Ryoma, et al.
Publicado: (2019)

Exploring the Role of Surfactants in Enhancing Drug Release from Amorphous Solid Dispersions at Higher Drug Loadings
por: Saboo, Sugandha, et al.
Publicado: (2021)

Role of Microstructure in Drug Release from Chitosan Amorphous Solid Dispersions
por: Lucio, David, et al.
Publicado: (2022)

A Comparative Study of the Pharmaceutical Properties between Amorphous Drugs Loaded-Mesoporous Silica and Pure Amorphous Drugs Prepared by Solvent Evaporation
por: Budiman, Arif, et al.
Publicado: (2022)

Combining drug salt formation with amorphous solid dispersions – a double edged sword
por: Hiew, Tze Ning, et al.
Publicado: (2022)

Amorphization of Thiamine Mononitrate: A Study of Crystallization Inhibition and Chemical Stability of Thiamine in Thiamine Mononitrate Amorphous Solid Dispersions
por: Arioglu-Tuncil, Seda, et al.
Publicado: (2020)

Amorphous Solid Dispersion of Epigallocatechin Gallate for Enhanced Physical Stability and Controlled Release
por: Cao, Yizheng, et al.
Publicado: (2017)

Cellulose based polymers in development of amorphous solid dispersions
por: Chavan, Rahul B, et al.
Publicado: (2019)

Preparation and Characterization of Amorphous Solid Dispersions for the Solubilization of Fenretinide
por: Zuccari, Guendalina, et al.
Publicado: (2023)

Amorphous Solid Dispersion as Drug Delivery Vehicles in Cancer
por: Budiman, Arif, et al.
Publicado: (2023)

Nilutamide
por: Trasi, Niraj S., et al.
Publicado: (2012)

Oral Delivery of Niclosamide as an Amorphous Solid Dispersion That Generates Amorphous Nanoparticles during Dissolution
por: Jara, Miguel O., et al.
Publicado: (2022)

Fed- and Fasted-State Performance of Pretomanid Amorphous Solid Dispersions Formulated with an Enteric Polymer
por: Nguyen, Hanh Thuy, et al.
Publicado: (2023)

Impact of Gastric pH Variations on the Release of Amorphous Solid Dispersion Formulations Containing a Weakly Basic Drug and Enteric Polymers
por: Nguyen, Hanh Thuy, et al.
Publicado: (2023)

Kinetics of Water-Induced Amorphous Phase Separation in Amorphous Solid Dispersions via Raman Mapping
por: Krummnow, Adrian, et al.
Publicado: (2023)

Preparation and Characterization of Spherical Amorphous Solid Dispersion with Amphotericin B
por: Mehenni, Lyes, et al.
Publicado: (2018)

Formulation Characterization and Pharmacokinetic Evaluation of Amorphous Solid Dispersions of Dasatinib
por: Dharani, Sathish, et al.
Publicado: (2022)

Stabilizing Mechanisms of β-Lactoglobulin in Amorphous Solid Dispersions of Indomethacin
por: Kabedev, Aleksei, et al.
Publicado: (2022)

Advances in the development of amorphous solid dispersions: The role of polymeric carriers
por: Zhang, Jie, et al.
Publicado: (2023)

Optimization of solid lipid nanoparticles prepared by a single emulsification-solvent evaporation method
por: Pooja, Deep, et al.
Publicado: (2015)

Enhancing the Solubility of Curcumin Using a Solid Dispersion System with Hydroxypropyl-β-Cyclodextrin Prepared by Grinding, Freeze-Drying, and Common Solvent Evaporation Methods
por: Mai, Nguyen Ngoc Sao, et al.
Publicado: (2020)

Enteric coating of tablets containing an amorphous solid dispersion of an enteric polymer and a weakly basic drug: A strategy to enhance in vitro release
por: Nguyen, Hanh Thuy, et al.
Publicado: (2023)

Bioavailability Improvement of Carbamazepine via Oral Administration of Modified-Release Amorphous Solid Dispersions in Rats
por: Li, Houli, et al.
Publicado: (2020)

Thermodynamic Modeling of the Amorphous Solid Dispersion-Water Interfacial Layer and Its Impact on the Release Mechanism
por: Dohrn, Stefanie, et al.
Publicado: (2023)

Microwave-Induced In Situ Amorphization: A New Strategy for Tackling the Stability Issue of Amorphous Solid Dispersions
por: Qiang, Wei, et al.
Publicado: (2020)

Amorphization of Thiamine Chloride Hydrochloride: Effects of Physical State and Polymer Type on the Chemical Stability of Thiamine in Solid Dispersions
por: Arioglu-Tuncil, Seda, et al.
Publicado: (2020)

Cannot write session to /tmp/vufind_sessions/sess_2dbi07eb7eojpqpl20ademqciu