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4-Nitrophenyl activated esters are superior synthons for indirect radiofluorination of biomolecules
Indirect radiolabelling has for a long time been the mainstay strategy for radiofluorination of biomolecules. Acylation of biomolecules through the use of an (18)F-labelled activated ester is a standard method for indirect radiolabelling. However, the preparation of (18)F-labelled activated esters i...
Autores principales: | Haskali, Mohammad B., Farnsworth, Ashleigh L., Roselt, Peter D., Hutton, Craig A. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Royal Society of Chemistry
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7517343/ https://www.ncbi.nlm.nih.gov/pubmed/33479687 http://dx.doi.org/10.1039/d0md00140f |
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