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Design, Synthesis and In Vitro Experimental Validation of Novel TRPV4 Antagonists Inspired by Labdane Diterpenes
Labdane diterpenes are widespread classes of natural compounds present in variety of marine and terrestrial organisms and plants. Many of them represents “natural libraries” of compounds with interesting biological activities due to differently functionalized drimane nucleus exploitable for potentia...
Autores principales: | Mazzotta, Sarah, Carullo, Gabriele, Schiano Moriello, Aniello, Amodeo, Pietro, Di Marzo, Vincenzo, Vega-Holm, Margarita, Vitale, Rosa Maria, Aiello, Francesca, Brizzi, Antonella, De Petrocellis, Luciano |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7594054/ https://www.ncbi.nlm.nih.gov/pubmed/33081023 http://dx.doi.org/10.3390/md18100519 |
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