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InhA inhibitors have activity against non-replicating Mycobacterium tuberculosis

We previously identified a diazaborine series with potential for development as a new tuberculosis drug. This series has activity in vitro and in vivo and targets cell wall biosynthesis via inhibition of InhA. The overall aim of this study was to determine whether InhA inhibitors have activity again...

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Detalles Bibliográficos
Autores principales: Flint, Lindsay, Korkegian, Aaron, Parish, Tanya
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Public Library of Science 2020
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7671525/
https://www.ncbi.nlm.nih.gov/pubmed/33201882
http://dx.doi.org/10.1371/journal.pone.0239354