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Novel 1-Amidino-4-Phenylpiperazines as Potent Agonists at Human TAAR1 Receptor: Rational Design, Synthesis, Biological Evaluation and Molecular Docking Studies

Targeting trace amine-associated receptor 1 (TAAR1) receptor continues to offer an intriguing opportunity to develop innovative therapies in different pharmacological settings. Pursuing our endeavors in the search for effective and safe human TAAR1 (hTAAR1) ligands, we synthesized a new series of 1-...

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Detalles Bibliográficos
Autores principales:	Francesconi, Valeria, Cichero, Elena, Kanov, Evgeny V., Laurini, Erik, Pricl, Sabrina, Gainetdinov, Raul R., Tonelli, Michele
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2020
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7697893/ https://www.ncbi.nlm.nih.gov/pubmed/33202687 http://dx.doi.org/10.3390/ph13110391

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