Cargando…

Synthesis and Biological Evaluation of Carvacrol-Based Derivatives as Dual Inhibitors of H. pylori Strains and AGS Cell Proliferation

This study reports on the synthesis, structural assessment, microbiological screening against several strains of H. pylori and antiproliferative activity against human gastric adenocarcinoma (AGS) cells of a large series of carvacrol-based compounds. Structural analyses consisted of elemental analys...

Descripción completa

Detalles Bibliográficos
Autores principales:	Sisto, Francesca, Carradori, Simone, Guglielmi, Paolo, Traversi, Carmen Beatrice, Spano, Mattia, Sobolev, Anatoly P., Secci, Daniela, Di Marcantonio, Maria Carmela, Haloci, Entela, Grande, Rossella, Mincione, Gabriella
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2020
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7699384/ https://www.ncbi.nlm.nih.gov/pubmed/33228095 http://dx.doi.org/10.3390/ph13110405

Ejemplares similares

Synthesis and Evaluation of Thymol-Based Synthetic Derivatives as Dual-Action Inhibitors against Different Strains of H. pylori and AGS Cell Line
por: Sisto, Francesca, et al.
Publicado: (2021)

Antimicrobial and Antibiofilm Activities of New Synthesized Silver Ultra-NanoClusters (SUNCs) Against Helicobacter pylori
por: Grande, Rossella, et al.
Publicado: (2020)

Identification and characterization of the α-CA in the outer membrane vesicles produced by Helicobacter pylori
por: Ronci, Maurizio, et al.
Publicado: (2019)

Antimicrobial and Antibiofilm Activities of Carvacrol, Amoxicillin and Salicylhydroxamic Acid Alone and in Combination vs. Helicobacter pylori: Towards a New Multi-Targeted Therapy
por: Puca, Valentina, et al.
Publicado: (2023)

Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents
por: Veschi, Serena, et al.
Publicado: (2020)

Eradication of Helicobacter pylori and Gastric Cancer: A Controversial Relationship
por: Piscione, Mariagrazia, et al.
Publicado: (2021)

The Antibiofilm Effect of a Medical Device Containing TIAB on Microorganisms Associated with Surgical Site Infection
por: Puca, Valentina, et al.
Publicado: (2019)

Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles
por: Grande, Rossella, et al.
Publicado: (2021)

Antibiofilm activity and NMR-based metabolomic characterization of cell-free supernatant of Limosilactobacillus reuteri DSM 17938
por: Vitale, Irene, et al.
Publicado: (2023)

In Vitro Activity of the Arylaminoartemisinin GC012 against Helicobacter pylori and Its Effects on Biofilm
por: Sisto, Francesca, et al.
Publicado: (2022)

Nature-Inspired Compounds: Synthesis and Antibacterial Susceptibility Testing of Eugenol Derivatives against H. pylori Strains
por: Carradori, Simone, et al.
Publicado: (2023)

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms
por: D’Ascenzio, Melissa, et al.
Publicado: (2016)

Helicobacter pylori ATCC 43629/NCTC 11639 Outer Membrane Vesicles (OMVs) from Biofilm and Planktonic Phase Associated with Extracellular DNA (eDNA)
por: Grande, Rossella, et al.
Publicado: (2015)

Effects of H(2)O(2) Treatment Combined With PI3K Inhibitor and MEK Inhibitor in AGS Cells: Oxidative Stress Outcomes in a Model of Gastric Cancer
por: Savino, Luca, et al.
Publicado: (2022)

Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Stationary Phase
por: Sadutto, Daniele, et al.
Publicado: (2023)

Carbonic Anhydrases: New Perspectives on Protein Functional Role and Inhibition in Helicobacter pylori
por: Campestre, Cristina, et al.
Publicado: (2021)

Carvacrol
por: Bogue, E. A.
Publicado: (1874)

PDAC, the Influencer Cancer: Cross-Talk with Tumor Microenvironment and Connected Potential Therapy Strategies
por: Mercanti, Leonardo, et al.
Publicado: (2023)

A Narrative Review on Non-Cirrohotic Portal Hypertension: Not All Portal Hypertensions Mean Cirrhosis
por: Fiordaliso, Michele, et al.
Publicado: (2023)

Novel Biologically Active Molecules, Biomaterials, and Nanoparticles for Microbial Biofilm Control in Human Medicine
por: Grande, Rossella, et al.
Publicado: (2021)

Doxorubicin-induced oxidative and nitrosative stress: Mitochondrial connexin 43 is at the crossroads
por: Pecoraro, Michela, et al.
Publicado: (2020)

Evaluation of In Vitro Capsaicin Release and Antimicrobial Properties of Topical Pharmaceutical Formulation
por: Goci, Enkelejda, et al.
Publicado: (2021)

The Beneficial Effect of Carvacrol in HL-1 Cardiomyocytes Treated with LPS-G: Anti-Inflammatory Pathway Investigations
por: Marconi, Guya Diletta, et al.
Publicado: (2022)

EGF and TGF-β1 Effects on Thyroid Function
por: Mincione, Gabriella, et al.
Publicado: (2011)

Potential Antibacterial Activity of Carvacrol-Loaded Poly(DL-lactide-co-glycolide) (PLGA) Nanoparticles against Microbial Biofilm
por: Iannitelli, Antonio, et al.
Publicado: (2011)

Editorial: Helicobacter pylori and its mechanisms of antibiotic survival
por: Krzyżek, Paweł, et al.
Publicado: (2023)

Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles
por: Guglielmi, Paolo, et al.
Publicado: (2019)

Alveolar Abscess.—Treatment with Carvacrol
por: Sage, H. L.
Publicado: (1875)

Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
por: Pontecorvi, Virginia, et al.
Publicado: (2022)

NMR-Based Approaches in the Study of Foods
por: Sobolev, Anatoly P., et al.
Publicado: (2022)

Detection and Physicochemical Characterization of Membrane Vesicles (MVs) of Lactobacillus reuteri DSM 17938
por: Grande, Rossella, et al.
Publicado: (2017)

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation
por: Guglielmi, Paolo, et al.
Publicado: (2020)

Open Questions in Cold Atmospheric Plasma Treatment in Head and Neck Cancer: A Systematic Review
por: Perrotti, Vittoria, et al.
Publicado: (2022)

Evaluation of SD BIOLINE H. pylori Ag rapid test against double ELISA with SD H. pylori Ag ELISA and EZ-STEP H. pylori Ag ELISA tests
por: Negash, Markos, et al.
Publicado: (2018)

Transformation of Helicobacter pylori into Coccoid Forms as a Challenge for Research Determining Activity of Antimicrobial Substances
por: Krzyżek, Paweł, et al.
Publicado: (2020)

Antifungal Carvacrol Loaded Chitosan Nanoparticles
por: Vitali, Alberto, et al.
Publicado: (2021)

Identification of the zinc finger 216 (ZNF216) in human carcinoma cells: a potential regulator of EGFR activity
por: Mincione, Gabriella, et al.
Publicado: (2016)

Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
por: Carradori, Simone, et al.
Publicado: (2017)

Correlation between the Antimicrobial Activity and Metabolic Profiles of Cell Free Supernatants and Membrane Vesicles Produced by Lactobacillus reuteri DSM 17938
por: Maccelli, Alessandro, et al.
Publicado: (2020)

Antimicrobial activity of essential oils and carvacrol, and synergy of carvacrol and erythromycin, against clinical, erythromycin-resistant Group A Streptococci
por: Magi, Gloria, et al.
Publicado: (2015)

Cannot write session to /tmp/vufind_sessions/sess_01lqgut7cer7a15kahdm07u0vc