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A General and Scalable Synthesis of Polysubstituted Indoles

A consecutive 2-step synthesis of N-unprotected polysubstituted indoles bearing an electron-withdrawing group at the C-3 position from readily available nitroarenes is reported. The protocol is based on the [3,3]-sigmatropic rearrangement of N-oxyenamines generated by the DABCO-catalyzed reaction of...

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Detalles Bibliográficos
Autores principales:	Tejedor, David, Diana-Rivero, Raquel, García-Tellado, Fernando
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2020
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7730962/ https://www.ncbi.nlm.nih.gov/pubmed/33260745 http://dx.doi.org/10.3390/molecules25235595

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