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New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives

In the present work, we report a new class of potent steroid sulphatase (STS) inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives. Within the set of new STS inhibitors, 6-(1-(1,2,3-trifluorophenyl)-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate 3L demonstra...

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Detalles Bibliográficos
Autores principales:	Ciupak, Olga, Daśko, Mateusz, Biernacki, Karol, Rachon, Janusz, Masłyk, Maciej, Kubiński, Konrad, Martyna, Aleksandra, Demkowicz, Sebastian
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2020
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7744152/ https://www.ncbi.nlm.nih.gov/pubmed/33322953 http://dx.doi.org/10.1080/14756366.2020.1858820

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