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Acylpolyamine Mygalin as a TLR4 Antagonist Based on Molecular Docking and In Vitro Analyses
Toll-like receptors (TLRs) are transmembrane proteins that are key regulators of innate and adaptive immune responses, particularly TLR4, and they have been identified as potential drug targets for the treatment of disease. Several low-molecular-weight compounds are being considered as new drug targ...
Autores principales: | Espinoza-Culupú, Abraham, Vázquez-Ramírez, Ricardo, Farfán-López, Mariella, Mendes, Elizabeth, Notomi Sato, Maria, da Silva Junior, Pedro Ismael, Borges, Monamaris Marques |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7761503/ https://www.ncbi.nlm.nih.gov/pubmed/33271940 http://dx.doi.org/10.3390/biom10121624 |
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