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Polypeptide-Based Molecular Platform and Its Docetaxel/Sulfo-Cy5-Containing Conjugate for Targeted Delivery to Prostate Specific Membrane Antigen
A strategy for stereoselective synthesis of molecular platform for targeted delivery of bimodal therapeutic or theranostic agents to the prostate-specific membrane antigen (PSMA) receptor was developed. The proposed platform contains a urea-based, PSMA-targeting Glu-Urea-Lys (EuK) fragment as a vect...
Autores principales: | Petrov, Stanislav A., Machulkin, Aleksei E., Uspenskaya, Anastasia A., Zyk, Nikolay Y., Nimenko, Ekaterina A., Garanina, Anastasia S., Petrov, Rostislav A., Polshakov, Vladimir I., Grishin, Yuri K., Roznyatovsky, Vitaly A., Zyk, Nikolay V., Majouga, Alexander G., Beloglazkina, Elena K. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7762530/ https://www.ncbi.nlm.nih.gov/pubmed/33302417 http://dx.doi.org/10.3390/molecules25245784 |
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