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The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification
We describe the assembly and annotation of a chemogenomic set of protein kinase inhibitors as an open science resource for studying kinase biology. The set only includes inhibitors that show potent kinase inhibition and a narrow spectrum of activity when screened across a large panel of kinase bioch...
Autores principales: | Wells, Carrow I., Al-Ali, Hassan, Andrews, David M., Asquith, Christopher R. M., Axtman, Alison D., Dikic, Ivan, Ebner, Daniel, Ettmayer, Peter, Fischer, Christian, Frederiksen, Mathias, Futrell, Robert E., Gray, Nathanael S., Hatch, Stephanie B., Knapp, Stefan, Lücking, Ulrich, Michaelides, Michael, Mills, Caitlin E., Müller, Susanne, Owen, Dafydd, Picado, Alfredo, Saikatendu, Kumar S., Schröder, Martin, Stolz, Alexandra, Tellechea, Mariana, Turunen, Brandon J., Vilar, Santiago, Wang, Jinhua, Zuercher, William J., Willson, Timothy M., Drewry, David H. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7826789/ https://www.ncbi.nlm.nih.gov/pubmed/33429995 http://dx.doi.org/10.3390/ijms22020566 |
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