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Structural Aspects of Photopharmacology: Insight into the Binding of Photoswitchable and Photocaged Inhibitors to the Glutamate Transporter Homologue
[Image: see text] Photopharmacology addresses the challenge of drug selectivity and side effects through creation of photoresponsive molecules activated with light with high spatiotemporal precision. This is achieved through incorporation of molecular photoswitches and photocages into the pharmacoph...
Autores principales: | Arkhipova, Valentina, Fu, Haigen, Hoorens, Mark W. H., Trinco, Gianluca, Lameijer, Lucien N., Marin, Egor, Feringa, Ben L., Poelarends, Gerrit J., Szymanski, Wiktor, Slotboom, Dirk J., Guskov, Albert |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2021
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7844824/ https://www.ncbi.nlm.nih.gov/pubmed/33449695 http://dx.doi.org/10.1021/jacs.0c11336 |
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