Cargando…

Structure, Function, and Pharmaceutical Ligands of 5-Hydroxytryptamine 2B Receptor

Since the first characterization of the 5-hydroxytryptamine 2B receptor (5-HT(2B)R) in 1992, significant progress has been made in 5-HT(2B)R research. Herein, we summarize the biological function, structure, and small-molecule pharmaceutical ligands of the 5-HT(2B)R. Emerging evidence has suggested...

Descripción completa

Detalles Bibliográficos
Autores principales:	Wang, Qing, Zhou, Yu, Huang, Jianhui, Huang, Niu
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Review
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7909583/ https://www.ncbi.nlm.nih.gov/pubmed/33498477 http://dx.doi.org/10.3390/ph14020076

Ejemplares similares

5- Hydroxytryptamine
por: Giarman, Nicholas J.
Publicado: (1958)

5-Hydroxytryptamine Receptor Subtypes and their Modulators with Therapeutic Potentials
por: Pithadia, Anand B., et al.
Publicado: (2009)

Serotonin in the rat prefrontal cortex controls the micturition reflex through 5‐hydroxytryptamine 2A and 5‐hydroxytryptamine 7 receptors
por: Chiba, Hiroki, et al.
Publicado: (2020)

5-Hydroxytryptamine Receptors and Tardive Dyskinesia in Schizophrenia
por: Pozhidaev, Ivan V., et al.
Publicado: (2020)

Remaining Need for In Vitro Test to Elucidate 5-Hydroxytryptamine 2C Receptor Functioning
por: Ivanova, Svetlana A., et al.
Publicado: (2018)

The 5-hydroxytryptamine 4 Receptor Agonist-induced Actions and Enteric Neurogenesis in the Gut
por: Takaki, Miyako, et al.
Publicado: (2014)

STORAGE OF 5-HYDROXYTRYPTAMINE IN MEGAKARYOCYTES
por: Tranzer, J. P., et al.
Publicado: (1972)

The Mechanism of Secretion and Metabolism of Gut-Derived 5-Hydroxytryptamine
por: Liu, Ning, et al.
Publicado: (2021)

Upregulation of 5-Hydroxytryptamine Receptor Signaling in Coronary Arteries after Organ Culture
por: Deng, Chun-Yu, et al.
Publicado: (2014)

Effective treatment with combination of peripheral 5‐hydroxytryptamine synthetic inhibitor and 5‐hydroxytryptamine 2 receptor antagonist on glucocorticoid‐induced whole‐body insulin resistance with hyperglycemia
por: Ma, Shaoxin, et al.
Publicado: (2016)

Structural Determinants of Ca(2+) Permeability and Conduction in the Human 5-Hydroxytryptamine Type 3A Receptor
por: Livesey, Matthew R., et al.
Publicado: (2008)

5-Hydroxytryptamine (serotonin) 2A receptor gene polymorphism is associated with schizophrenia
por: Sujitha, Subash Padmajeya, et al.
Publicado: (2014)

Involvement of 5-Hydroxytryptamine Receptor 2A in the Pathophysiology of Medication-Overuse Headache
por: Zheng, Zhenyang, et al.
Publicado: (2021)

Dynamics and Patterning of 5-Hydroxytryptamine 2 Subtype Receptors in JC Polyomavirus Entry
por: Mehmood, Kashif, et al.
Publicado: (2022)

Possible Role of 5-Hydroxytryptamine (5-HT) Receptor on Human Sperm Motility Regulation
por: Omote, Maya, et al.
Publicado: (2023)

Phylogenetic analyses of 5-hydroxytryptamine 3 (5-HT(3)) receptors in Metazoa
por: Rao, Santosh T. R. B., et al.
Publicado: (2023)

Association of 5-Hydroxytryptamine 3 Receptor Antagonists With the Prognosis of Liver Failure
por: Chen, Yuting, et al.
Publicado: (2021)

A Meta-Analysis of 5-Hydroxytryptamine Receptor 1B Polymorphisms With Risk of Major Depressive Disorder and Suicidal Behavior
por: Yang, Pingliang, et al.
Publicado: (2021)

Anxiety-induced hyperalgesia in female rats is mediated by cholecystokinin 2 receptor in rostral ventromedial medulla and spinal 5-hydroxytryptamine 2B receptor
por: Jiang, Ming, et al.
Publicado: (2019)

Development of Plate Reader and On-Line Microfluidic Screening to Identify Ligands of the 5-Hydroxytryptamine Binding Protein in Venoms
por: Otvos, Reka A., et al.
Publicado: (2015)

The Effect of 5-Hydroxytryptamine Receptor Antagonist in Preventing Pain/Limb Shrinkage Reaction Associated with Rocuronium Injection
por: He, Qixiong, et al.
Publicado: (2018)

Inhibiting 5-hydroxytryptamine receptor 3 alleviates pathological changes of a mouse model of Alzheimer’s disease
por: Liu, Li-Fen, et al.
Publicado: (2023)

Structure–Activity Relationship and Evaluation of Phenethylamine and Tryptamine Derivatives for Affinity towards 5-Hydroxytryptamine Type 2A Receptor
por: Wang, Shujie, et al.
Publicado: (2023)

The anti-emetic potential of the 5-hydroxytryptamine3 receptor antagonist BRL 43694.
por: Bermudez, J., et al.
Publicado: (1988)

The 5‐hydroxytryptamine(4) receptor enables differentiation of informational content and encoding in the hippocampus
por: Twarkowski, Hannah, et al.
Publicado: (2016)

Potential Clinical Value of 5-Hydroxytryptamine Receptor 3C as a Prognostic Biomarker for Lung Cancer
por: Chen, Jiun-Rung, et al.
Publicado: (2021)

Structural Modification of the Antidepressant Mianserin Suggests That Its Anti-inflammatory Activity May Be Independent of 5-Hydroxytryptamine Receptors
por: Sacre, Sandra, et al.
Publicado: (2019)

Physiological Control of Molluscan Gill Cilia by 5-Hydroxytryptamine
por: Gosselin, R. E., et al.
Publicado: (1962)

CHEMICAL AND ULTRASTRUCTURAL IDENTIFICATION OF 5-HYDROXYTRYPTAMINE IN AN IDENTIFIED NEURON
por: Rude, Sonia, et al.
Publicado: (1969)

Neuroprotection by 2,3,5,4ʹ-tetrahydroxystilbene-2-O-β-D-glucoside extracts from Polygonum multiflorum against cerebral ischemia/reperfusion injury through the 5-hydroxytryptamine/5-hydroxytryptamine receptor pathway
por: Yi, Chuan-An, et al.
Publicado: (2019)

Evidence that 5-hydroxytryptamine3 receptors mediate cytotoxic drug and radiation-evoked emesis.
por: Miner, W. D., et al.
Publicado: (1987)

Lasmiditan and 5-Hydroxytryptamine in the rat trigeminal system; expression, release and interactions with 5-HT(1) receptors
por: Edvinsson, Jacob C. A., et al.
Publicado: (2022)

Blockade of 5-Hydroxytryptamine 2A Receptor Attenuates Precipitation of Naloxone-Induced Withdrawal Symptoms in Opioid-Exposed Mice
por: Li, Bing, et al.
Publicado: (2022)

Potentiation of RSU-1069 tumour cytotoxicity by 5-hydroxytryptamine (5-HT).
por: Chaplin, D. J.
Publicado: (1986)

The Relationship Between 5-Hydroxytryptamine and Its Metabolite Changes With Post-stroke Depression
por: Gu, Simeng, et al.
Publicado: (2022)

Bilirubin Induces Pain Desensitization in Cholestasis by Activating 5-Hydroxytryptamine 3A Receptor in Spinal Cord
por: Kong, Erliang, et al.
Publicado: (2021)

UFLC-PDA-MS/MS Profiling of Seven Uncaria Species Integrated with Melatonin/5-Hydroxytryptamine Receptors Agonistic Assay
por: Zhang, Jian-Gang, et al.
Publicado: (2020)

Two cases of mild serotonin toxicity via 5-hydroxytryptamine 1A receptor stimulation
por: Nakayama, Hiroto, et al.
Publicado: (2014)

The impact of 5-hydroxytryptamine-receptor antagonists on chemotherapy treatment adherence, treatment delay, and nausea and vomiting
por: Palli, Swetha Rao, et al.
Publicado: (2015)

Tricyclic antidepressant amitriptyline inhibits 5-hydroxytryptamine 3 receptor currents in NCB-20 cells
por: Park, Yong Soo, et al.
Publicado: (2018)

Cannot write session to /tmp/vufind_sessions/sess_0g7asqgbcra5alk05m1rivha2l