Cargando…

Easy-To-Access Quinolone Derivatives Exhibiting Antibacterial and Anti-Parasitic Activities

The cell wall of Mycobacterium tuberculosis (Mtb) has a unique structural organisation, comprising a high lipid content mixed with polysaccharides. This makes cell wall a formidable barrier impermeable to hydrophilic agents. In addition, during host infection, Mtb resides in macrophages within avasc...

Descripción completa

Detalles Bibliográficos
Autores principales:	Beteck, Richard M., Jordaan, Audrey, Seldon, Ronnett, Laming, Dustin, Hoppe, Heinrich C., Warner, Digby F., Khanye, Setshaba D.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7931078/ https://www.ncbi.nlm.nih.gov/pubmed/33672753 http://dx.doi.org/10.3390/molecules26041141

Ejemplares similares

New Quinolone-Based Thiosemicarbazones Showing Activity Against Plasmodium falciparum and Mycobacterium tuberculosis
por: Beteck, Richard M., et al.
Publicado: (2019)

Cinnamoyl-Oxaborole Amides: Synthesis and Their in Vitro Biological Activity
por: Gumbo, Maureen, et al.
Publicado: (2018)

Anti-Trypanosomal and Antimalarial Properties of Tetralone Derivatives and Structurally Related Benzocycloalkanones
por: Beteck, Richard M., et al.
Publicado: (2019)

Quinolone-3-amidoalkanol: A New Class of Potent and Broad-Spectrum Antimicrobial Agent
por: Dube, Phelelisiwe S., et al.
Publicado: (2023)

Biological Profiling Enables Rapid Mechanistic Classification of Phenotypic Screening Hits and Identification of KatG Activation-Dependent Pyridine Carboxamide Prodrugs With Activity Against Mycobacterium tuberculosis
por: Chengalroyen, Melissa D., et al.
Publicado: (2020)

Identification of Antimycobacterial Natural Products from a Library of Marine Invertebrate Extracts
por: Acquah, Kojo Sekyi, et al.
Publicado: (2022)

Coumarin-Annulated Ferrocenyl 1,3-Oxazine Derivatives Possessing In Vitro Antimalarial and Antitrypanosomal Potency
por: Mbaba, Mziyanda, et al.
Publicado: (2021)

Antimycobacterial Activity, Synergism, and Mechanism of Action Evaluation of Novel Polycyclic Amines against Mycobacterium tuberculosis
por: Kapp, Erika, et al.
Publicado: (2021)

Exploration of 4-aminopyrrolo[2,3-d]pyrimidine as antitubercular agents
por: Jesumoroti, Omobolanle Janet, et al.
Publicado: (2022)

Quinolone: a versatile therapeutic compound class
por: Dube, Phelelisiwe S., et al.
Publicado: (2022)

Aerosolization of Mycobacterium tuberculosis by Tidal Breathing
por: Dinkele, Ryan, et al.
Publicado: (2020)

Recent progress in the development of anti-malarial quinolones
por: Beteck, Richard M, et al.
Publicado: (2014)

Synthesis, Structure and In Vitro Anti-Trypanosomal Activity of Non-Toxic Arylpyrrole-Based Chalcone Derivatives
por: Zulu, Ayanda I., et al.
Publicado: (2020)

Discovery of Novel Thiazolidinedione-Derivatives with Multi-Modal Antidiabetic Activities In Vitro and In Silico
por: Arineitwe, Charles, et al.
Publicado: (2023)

Identification of Novel Potential Inhibitors of Pteridine Reductase 1 in Trypanosoma brucei via Computational Structure-Based Approaches and in Vitro Inhibition Assays
por: Kimuda, Magambo Phillip, et al.
Publicado: (2019)

The Current Case of Quinolones: Synthetic Approaches and Antibacterial Activity
por: Naeem, Abdul, et al.
Publicado: (2016)

A “Double-Edged” Scaffold: Antitumor Power within the  Antibacterial Quinolone
por: Bisacchi, Gregory S., et al.
Publicado: (2016)

Essential Guide of Analysis Methods Applied to Silver Complexes with Antibacterial Quinolones
por: Rusu, Aura, et al.
Publicado: (2018)

Structural Characterization of the Millennial Antibacterial (Fluoro)Quinolones—Shaping the Fifth Generation
por: Rusu, Aura, et al.
Publicado: (2021)

Surface-Growing Communities of Pseudomonas aeruginosa Exhibit Distinct Alkyl Quinolone Signatures
por: Morales-Soto, Nydia, et al.
Publicado: (2018)

Easy access to antifungal agents.
por: Faro, S
Publicado: (1999)

Easy Access to Evans’ Oxazolidinones. Stereoselective Synthesis and Antibacterial Activity of a New 2-Oxazolidinone Derivative
por: Diaz, Gaspar, et al.
Publicado: (2014)

A19 The impact of HIV-1 on the evolution of Mycobacterium tuberculosis
por: Koch, Anastasia, et al.
Publicado: (2018)

The Influence of HIV on the Evolution of Mycobacterium tuberculosis
por: Koch, Anastasia S., et al.
Publicado: (2017)

Structural basis for the inhibition of RecBCD by Gam and its synergistic antibacterial effect with quinolones
por: Wilkinson, Martin, et al.
Publicado: (2016)

Easy Access to Polyfunctionalized Chiral Decalins
por: Santalla, Hugo, et al.
Publicado: (2020)

Quinolone Allergy
por: McGee, Edoabasi U., et al.
Publicado: (2019)

Quinolone antibiotics
por: Pham, Thu D. M., et al.
Publicado: (2019)

Antimycobacterial, Cytotoxic, and Antioxidant Activities of Abietane Diterpenoids Isolated from Plectranthus madagascariensis
por: Ndjoubi, Kadidiatou O., et al.
Publicado: (2021)

CID12261165, a flavonoid compound as antibacterial agents against quinolone-resistant Staphylococcus aureus
por: Morimoto, Yuh, et al.
Publicado: (2023)

Synthesis of Quinolones and Zwitterionic Quinolonate Derivatives with Broad-Spectrum Antibiotic Activity
por: Suay-García, Beatriz, et al.
Publicado: (2022)

UREKA: Umbilical Ring Easy Kannula Access
por: Carlson, Jared W., et al.
Publicado: (2011)

Easy Access to Phosphine‐Borane Building Blocks
por: de Jong, G. Bas, et al.
Publicado: (2020)

An Easy Access to Furan-Fused Polyheterocyclic Systems
por: Benzi, Alice, et al.
Publicado: (2022)

Quinolone Safety and Efficacy
por: Bellomo, Spartaco
Publicado: (2005)

Physicochemical Studies and Anticancer Potency of Ruthenium η(6)-p-Cymene Complexes Containing Antibacterial Quinolones
por: Kljun, Jakob, et al.
Publicado: (2011)

In Vitro and In Vivo Antibacterial Activities of a Novel Quinolone Compound, OPS-2071, against Clostridioides difficile
por: Oka, Daisuke, et al.
Publicado: (2021)

Detection of the in vitro modulation of Plasmodium falciparum Arf1 by Sec7 and ArfGAP domains using a colorimetric plate-based assay
por: Swart, Tarryn, et al.
Publicado: (2020)

Quinolone Resistance in Gallibacterium anatis Determined by Mutations in Quinolone Resistance-Determining Region
por: Rømer Villumsen, Kasper, et al.
Publicado: (2023)

Endochin-Like Quinolones Exhibit Promising Efficacy Against Neospora Caninum in vitro and in Experimentally Infected Pregnant Mice
por: Anghel, Nicoleta, et al.
Publicado: (2018)

Cannot write session to /tmp/vufind_sessions/sess_5b61hqq4k1rhb3td9htc25l8m4