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Development of a ghrelin receptor inverse agonist for positron emission tomography
Imaging of Ghrelin receptors in vivo provides unique potential to gain deeper understanding on Ghrelin and its receptors in health and disease, in particular, in cancer. Ghrelin, an octanoylated 28-mer peptide hormone activates the constitutively active growth hormone secretagogue receptor type 1a (...
Autores principales: | Bergmann, Ralf, Chollet, Constance, Els-Heindl, Sylvia, Ullrich, Martin, Berndt, Nicole, Pietzsch, Jens, Máthé, Domokos, Bachmann, Michael, Beck-Sickinger, Annette G. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Impact Journals LLC
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7939532/ https://www.ncbi.nlm.nih.gov/pubmed/33747360 http://dx.doi.org/10.18632/oncotarget.27895 |
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