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A Systematic Study of the In Vitro Pharmacokinetics and Estimated Human In Vivo Clearance of Indole and Indazole-3-Carboxamide Synthetic Cannabinoid Receptor Agonists Detected on the Illicit Drug Market
In vitro pharmacokinetic studies were conducted on enantiomer pairs of twelve valinate or tert-leucinate indole and indazole-3-carboxamide synthetic cannabinoid receptor agonists (SCRAs) detected on the illicit drug market to investigate their physicochemical parameters and structure-metabolism rela...
Autores principales: | Brandon, Andrew M., Antonides, Lysbeth H., Riley, Jennifer, Epemolu, Ola, McKeown, Denise A., Read, Kevin D., McKenzie, Craig |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7961380/ https://www.ncbi.nlm.nih.gov/pubmed/33807614 http://dx.doi.org/10.3390/molecules26051396 |
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