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The Open Question of How GPCRs Interact with GPCR Kinases (GRKs)
G protein-coupled receptors (GPCRs), which regulate a vast number of eukaryotic processes, are desensitized by various mechanisms but, most importantly, by the GPCR kinases (GRKs). Ever since GRKs were first identified, investigators have sought to determine which structural features of GRKs are use...
Autores principales: | Cato, M. Claire, Yen, Yu-Chen, Francis, Charnelle J., Elkins, Kaely E., Shareef, Afzaal, Sterne-Marr, Rachel, Tesmer, John J. G. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8002388/ https://www.ncbi.nlm.nih.gov/pubmed/33802765 http://dx.doi.org/10.3390/biom11030447 |
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