Cargando…

The Antitumor Peptide ERα17p Exerts Anti-Hyperalgesic and Anti-Inflammatory Actions Through GPER in Mice

Persistent inflammation and persistent pain are major medical, social and economic burdens. As such, related pharmacotherapy needs to be continuously improved. The peptide ERα17p, which originates from a part of the hinge region/AF2 domain of the human estrogen receptor α (ERα), exerts anti-prolifer...

Descripción completa

Detalles Bibliográficos
Autores principales:	Mallet, Christophe, Boudieu, Ludivine, Lamoine, Sylvain, Coudert, Catherine, Jacquot, Yves, Eschalier, Alain
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Frontiers Media S.A. 2021
Materias:	Endocrinology
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8011567/ https://www.ncbi.nlm.nih.gov/pubmed/33815268 http://dx.doi.org/10.3389/fendo.2021.578250

Ejemplares similares

The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells
por: Lappano, Rosamaria, et al.
Publicado: (2019)

Deciphering of a Putative GPER Recognition Domain in ERα and ERα36
por: Acramel, Alexandre, et al.
Publicado: (2022)

Anti-Hyperalgesic Properties of Menthol and Pulegone
por: Hilfiger, Louis, et al.
Publicado: (2021)

Promising Perspectives of the Antiproliferative GPER Inverse Agonist ERα17p in Breast Cancer
por: Kampa, Marilena, et al.
Publicado: (2023)

Interaction of the Anti-Proliferative GPER Inverse Agonist ERα17p with the Breast Cancer Cell Plasma Membrane: From Biophysics to Biology
por: Trichet, Michaël, et al.
Publicado: (2020)

GPER1 Activation Exerts Anti-Tumor Activity in Multiple Myeloma
por: Gallo Cantafio, Maria Eugenia, et al.
Publicado: (2023)

Editorial: GPER and Human Pathologies
por: Jacquot, Yves, et al.
Publicado: (2021)

Editorial: GPER: Control and Functions
por: Jacquot, Yves, et al.
Publicado: (2021)

Anti-inflammatory and anti-hyperalgesic activities of Acanthopanax trifoliatus (L) Merr leaves
por: Hamid, Roslida Abdul, et al.
Publicado: (2013)

The Importance of Perioperative Administration of an Anti-Hyperalgesic Drug in Burn Wounds
por: Dalle Carbonare, Luca, et al.
Publicado: (2012)

Anti-hyperalgesic effects of calcitonin on neuropathic pain interacting with its peripheral receptors
por: Ito, Akitoshi, et al.
Publicado: (2012)

Oral Ultramicronized Palmitoylethanolamide: Plasma and Tissue Levels and Spinal Anti-hyperalgesic Effect
por: Petrosino, Stefania, et al.
Publicado: (2018)

Computational Approaches for the Discovery of GPER Targeting Compounds
por: Grande, Fedora, et al.
Publicado: (2020)

Identification of a human estrogen receptor α tetrapeptidic fragment with dual antiproliferative and anti-nociceptive action
por: Jouffre, Baptiste, et al.
Publicado: (2023)

Minocycline potentiates the anti-hyperalgesic effect of ceftriaxone in CCI-induced neuropathic pain in rats
por: Amin, B., et al.
Publicado: (2015)

Hyperalgesic activity of kisspeptin in mice
por: Spampinato, Simona, et al.
Publicado: (2011)

The Class I HDAC Inhibitor, MS-275, Prevents Oxaliplatin-Induced Chronic Neuropathy and Potentiates Its Antiproliferative Activity in Mice
por: Lamoine, Sylvain, et al.
Publicado: (2021)

Potentiation of Amitriptyline Anti-Hyperalgesic-Like Action By Astroglial Connexin 43 Inhibition in Neuropathic Rats
por: Jeanson, Tiffany, et al.
Publicado: (2016)

Estrogen Signaling in ERα-Negative Breast Cancer: ERβ and GPER
por: Girgert, Rainer, et al.
Publicado: (2019)

NHERF1, a novel GPER associated protein, increases stability and activation of GPER in ER-positive breast cancer
por: Meng, Ran, et al.
Publicado: (2016)

Anti-hyperalgesic properties of a flavanone derivative Poncirin in acute and chronic inflammatory pain models in mice
por: Afridi, Ruqayya, et al.
Publicado: (2019)

The Co-Expression of Estrogen Receptors ERα, ERβ, and GPER in Endometrial Cancer
por: Hojnik, Marko, et al.
Publicado: (2023)

Anti-allodynic and Anti-hyperalgesic effects of an ethanolic extract and xylopic acid from the fruits of Xylopia aethiopica in murine models of neuropathic pain
por: Ameyaw, Elvis O., et al.
Publicado: (2014)

Anti-hyperalgesic effects of a novel TRPM8 agonist in neuropathic rats: A comparison with topical menthol
por: Patel, Ryan, et al.
Publicado: (2014)

Neuroendocrine mechanisms in oxaliplatin-induced hyperalgesic priming
por: Staurengo-Ferrari, Larissa, et al.
Publicado: (2023)

Evaluation of Anti-Hyperalgesic and Analgesic Effects of Two Benzodiazepines in Human Experimental Pain: A Randomized Placebo-Controlled Study
por: Vuilleumier, Pascal H., et al.
Publicado: (2013)

Retraction Note: Anti-hyperalgesic properties of a flavanone derivative Poncirin in acute and chronic inflammatory pain models in mice
por: Afridi, Ruqayya, et al.
Publicado: (2023)

GPER expressed on microglia mediates the anti‐inflammatory effect of estradiol in ischemic stroke
por: Zhao, Tian‐Zhi, et al.
Publicado: (2016)

An Updated Review on the Metabolite (AM404)-Mediated Central Mechanism of Action of Paracetamol (Acetaminophen): Experimental Evidence and Potential Clinical Impact
por: Mallet, Christophe, et al.
Publicado: (2023)

Pretreatment with intrathecal amitriptyline potentiates anti-hyperalgesic effects of post-injury intra-peritoneal amitriptyline following spinal nerve ligation
por: Cheng, Kuang-I, et al.
Publicado: (2012)

Transcription factor Sp4 is required for hyperalgesic state persistence
por: Sheehan, Kayla, et al.
Publicado: (2019)

Lectin from Crataeva tapia bark exerts antitumor, anti-inflammtory and analgesic activities
por: Araújo, Regina M. S., et al.
Publicado: (2011)

Anti-hyperalgesic effects of photobiomodulation therapy (904 nm) on streptozotocin-induced diabetic neuropathy imply MAPK pathway and calcium dynamics modulation
por: Vieira, Willians Fernando, et al.
Publicado: (2022)

Assessment of the Anti-Allodynic and Anti-Hyperalgesic Efficacy of a Glycine Transporter 2 Inhibitor Relative to Pregabalin, Duloxetine and Indomethacin in a Rat Model of Cisplatin-Induced Peripheral Neuropathy
por: Kuo, Andy, et al.
Publicado: (2021)

LBODP005 Gper Modulates Multiple Functions In Adipose Tissue To Promote An Anti-obese Phenotype
por: Sharma, Geetanjali, et al.
Publicado: (2022)

Bazi Bushen Capsule Alleviates Post-Menopausal Atherosclerosis via GPER1-Dependent Anti-Inflammatory and Anti-Apoptotic Effects
por: Huang, Dan, et al.
Publicado: (2021)

Evidence for the Involvement of Spinal Cord-Inhibitory and Cytokines-Modulatory Mechanisms in the Anti-Hyperalgesic Effect of Hecogenin Acetate, a Steroidal Sapogenin-Acetylated, in Mice
por: Quintans, Jullyana S.S., et al.
Publicado: (2014)

Anti-Hyperalgesic Efficacy of Acetyl L-Carnitine (ALCAR) Against Visceral Pain Induced by Colitis: Involvement of Glia in the Enteric and Central Nervous System
por: Lucarini, Elena, et al.
Publicado: (2023)

Neurocognitive evidence for mental imagery-driven hypoalgesic and hyperalgesic pain regulation
por: Fardo, Francesca, et al.
Publicado: (2015)

Store‐operated calcium entry mediates hyperalgesic responses during neuropathy
por: Wang, Wei, et al.
Publicado: (2023)

Cannot write session to /tmp/vufind_sessions/sess_r76ag4hu8s6ck0cvc84cn44m6u