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1,2,4-Oxadiazole-Bearing Pyrazoles as Metabolically Stable Modulators of Store-Operated Calcium Entry

[Image: see text] Store-operated calcium entry (SOCE) is a pivotal mechanism in calcium homeostasis, and, despite still being under investigation, its dysregulation is known to be associated with severe human disorders. SOCE modulators are therefore needed both as chemical probes and as therapeutic...

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Detalles Bibliográficos
Autores principales:	Aprile, Silvio, Riva, Beatrice, Bhela, Irene Preet, Cordero-Sanchez, Celia, Avino, Giulia, Genazzani, Armando A., Serafini, Marta, Pirali, Tracey
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2021
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8040252/ https://www.ncbi.nlm.nih.gov/pubmed/33854704 http://dx.doi.org/10.1021/acsmedchemlett.1c00034

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