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A Pd-Catalyzed [4 + 2] Annulation Approach to Fluorinated N-Heterocycles
[Image: see text] 3-Fluoro- and trifluoromethylthio-piperidines represent important building blocks for discovery chemistry. We report a simple and efficient method to access analogs of these compounds that are armed with rich functionality allowing them to be chemoselectively derivatized with high...
Autores principales: | García-Vázquez, Víctor, Hoteite, Larry, Lakeland, Christopher P., Watson, David W., Harrity, Joseph P. A. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2021
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8041373/ https://www.ncbi.nlm.nih.gov/pubmed/33759534 http://dx.doi.org/10.1021/acs.orglett.1c00752 |
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